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N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
N-ethyl-3-(4-fluorophenyl)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)propanamide
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
8-(naphthalen-2-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidine-2,6-dione
N-(2,5-dimethoxyphenyl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-(methoxymethyl)pyrimidine
2-amino-7-(quinoline-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-({2-amino-6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
2-[ethyl(methyl)amino]-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[1-(2-fluorophenyl)propan-2-yl]-1,4-diazepan-5-one
ethyl[(6-methoxypyridin-3-yl)methyl][2-(1H-pyrazol-1-yl)ethyl]amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[1-({1-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}piperidin-2-one
(3aS,6aS)-5-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methyl-5-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-1,3-thiazol-2-amine
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(5-phenyl-1,3,4-thiadiazol-2-yl)urea
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-propoxypiperidine
1-[(3-fluorophenyl)methyl]-4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
3-(4-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
2-(5-acetylthiophen-3-yl)-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
8-(5-chloropyridine-2-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N3-cyclohexyl-1-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(2R,4R)-N-(9H-fluoren-9-yl)-4-hydroxypyrrolidine-2-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyrimidin-4-ol
N-{2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
3-{1-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
1-[(3-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-5-(morpholine-4-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[2-(methylsulfanyl)ethyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 6-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)pyridine-2-carboxylate
3-(2-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-3,4-dihydro-1,2,3-benzotriazin-4-one
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(pyrrolidin-1-yl)acetamide
4-[(2-butyl-1H-imidazol-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-({5-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
4-(4-chlorophenyl)-N-(2,2,2-trifluoroethyl)butanamide
2-(1H-imidazol-1-yl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]acetamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-methylpyrimidin-4-amine
4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}thiomorpholine
8-fluoro-2-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}quinoline
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(1H-indazole-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine
2-methoxy-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]pyridine
methyl[(2E)-3-phenylprop-2-en-1-yl](4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
3-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}sulfonyl)pyridine
5-chloro-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}thiophene-2-sulfonamide