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4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(3-methylphenyl)methyl]piperidin-4-ol
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
1-[(1S,5R)-6-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-[3-(trifluoromethyl)piperidin-1-yl]pyridine-3-carboxamide
4-phenyl-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine
{1,3-bis[(2-methylphenyl)methyl]piperidin-3-yl}methanol
2-phenyl-5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
1-ethyl-1-(oxan-2-ylmethyl)-3-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
2-(2,5-dioxoimidazolidin-4-yl)-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}acetamide
(1R,5S)-6-({5-[(2-ethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-6-azabicyclo[3.2.1]octane
2-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)-1,2-oxazolidine
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
3-(3-methoxypropyl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-3-carboxylic acid
3-(4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}phenyl)prop-2-yn-1-ol
4-[6-(methoxymethyl)pyrimidin-4-yl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-(2-methoxyphenyl)pyridazin-3-amine
3-(4-chloro-2-methylbenzoyl)-1-cyclobutylpiperidine
ethyl 1-[(2-chloro-4-fluorophenyl)methyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-5-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]pyridine-4-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(1H-indol-3-yl)butan-1-one
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-oxobutanamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4-fluorophenoxy)piperidine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[(1S)-1-phenylethyl]-1H-pyrazole-3-carboxamide
methyl 2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]pyridine-3-carboxylate
N,2-dimethyl-3-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-9-methyl-9H-carbazole
2-(2-methoxyethoxy)-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
(3S,4R)-1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[2-fluoro-5-({[3-(4-methyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)phenyl]-2-methylpropanamide
3-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(thiophen-2-yl)-1H-imidazole
5-acetyl-6-methyl-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]acetamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(furan-2-ylmethyl)piperidine
2-ethyl-N,4-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-oxazole-5-carboxamide
dimethyl(2-{2-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
5-butyl-1-(3-chlorophenyl)-4-(pyridazine-3-carbonyl)piperazin-2-one
6-(4-ethylphenyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
N-[3-(1H-indol-2-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
N3-tert-butyl-1-cyclohexyl-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-({4-[3-(2,5-dihydro-1H-pyrrole-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]azepan-4-amine