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5-(2-chloro-4-methoxyphenoxymethyl)-3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
N-{1-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]pyrrolidin-3-yl}acetamide
1-(5-chloro-2-methoxyphenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-(morpholin-2-yl)ethan-1-one
4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}morpholine-2-carboxylic acid
(2S,4S)-4-amino-1-(3-methoxybenzenesulfonyl)-N-methylpyrrolidine-2-carboxamide
3-{2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)acetamide
(1R,6S)-3-(1-benzyl-1H-pyrazole-4-carbonyl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(3-fluorophenyl)methyl]-1-methylpiperidine-2-carboxamide
2-(cyclopropylmethyl)-7-methyl-N-[(4-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(3-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
1-(furan-2-carbonyl)-4-{2-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}piperidine
6-(2,5-dimethylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-3-carboxamide
N-(propan-2-yl)-2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]acetamide
1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}cyclobutanamine
3-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-[(4-methoxyphenyl)methyl]propanamide
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-phenylpiperazine
5-(2-methylpropyl)-1'-(1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(2-methylpropyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-5-carboxamide
1-(2-chloropyridin-3-yl)-3-[1-(methoxymethyl)cyclopentyl]urea
(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)urea
5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-4-methylpyrimidin-2-amine
4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}benzoic acid
ethyl 4-(2-phenylethyl)-1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylate
4-acetamido-N,2-dimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
N-(4-methoxy-2-methylphenyl)-3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}propanamide
6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-9H-purin-2-amine
methyl[(4-methyl-1H-imidazol-5-yl)methyl][(5-propyl-1H-pyrazol-3-yl)methyl]amine
3-(2H-1,3-benzodioxol-5-yl)-5-(5-methoxyfuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-{3-[2-(2-methoxyethyl)morpholine-4-carbonyl]phenyl}-2-methylbutan-2-ol
2-methyl-3-{3-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]phenyl}pyrazine
(1R,5S)-6-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
8-(dimethyl-1,2-oxazole-4-carbonyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-hydroxyethyl)-2,6-dimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-4-carboxamide
(1-{[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
3-{[4-(3-chlorophenyl)-5-{[(cyclohex-3-en-1-ylmethyl)(methyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}benzonitrile
(1S,5R)-3-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-methyl-2-(3-propoxyphenyl)pyridine-4-carboxamide
2-[benzyl({4-[4-(furan-2-carbonyl)piperazin-1-yl]quinazolin-2-yl}methyl)amino]ethan-1-ol
2-hydroxy-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]acetamide
2-{1-[3-(azepan-1-ylmethyl)benzoyl]piperidin-2-yl}acetamide
5-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-4-(morpholin-4-yl)-N-(oxolan-2-ylmethyl)benzamide
5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N-phenylpyrimidin-2-amine