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8-[(2-aminopyridin-3-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-cyclohexyl-N-(cyclopropylmethyl)-3-(3-hydroxy-3-methylbutyl)benzamide
1-[(3-fluorophenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)piperidine-3-carboxamide
methyl 5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(4aS,8aR)-1-(3-aminopropyl)-6-(2-fluorobenzoyl)-decahydro-1,6-naphthyridin-2-one
methyl 3-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}benzamide
N,N-dimethyl-6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazin-2-amine
(3R,9R)-11-[4-(trifluoromethoxy)benzoyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
2-methyl-1,3-dioxo-N-(thiolan-3-yl)-2,3-dihydro-1H-isoindole-5-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-3-fluoro-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
1-[(3-methoxyphenyl)methyl]-4-[4-(pyridin-4-yl)pyrimidin-2-yl]piperazin-2-one
2-chloro-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)benzamide
N-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(morpholin-4-yl)acetamide
N-ethyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-(pyridin-4-ylmethyl)propanamide
(2R)-2-amino-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
(5S,9aS,9bS)-2-cyclopentyl-5-(2,4-dimethoxy-3-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-({1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-3-yl}methyl)benzoic acid
(2S)-2-[3-(4-chlorophenyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
3-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1-phenylurea
N-(1-benzylpyrrolidin-3-yl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}propanamide
(3R,9aR)-8-benzoyl-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}acetamide
1-(4-ethenylbenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
N-[(3S,4R)-4-propyl-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanesulfonamide
[3-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]methanol
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazole
2-(adamantan-1-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
2-methyl-8-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2,8-diazaspiro[4.5]decane
1-(2-aminoethyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
2-(3-methoxypropyl)-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methoxypyridine-4-carbonyl)pyrrolidine-3-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(cyclohexylmethyl)acetamide
2-ethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)pyrimidine-5-carboxamide
1-{4-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]phenyl}-3-(thiolan-3-yl)urea
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-amino-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyridine-2-carboxamide
2-(benzyloxy)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one
(3aR,6aR)-2-methanesulfonyl-5-[(2-methylpyrimidin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-aminopropanoyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
6-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-3-ol
N-(2-methyl-1-{7-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)oxolane-3-carboxamide
2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
3-cyclopropyl-1-[3-(methylsulfamoyl)phenyl]-3-[(3-methylthiophen-2-yl)methyl]urea
(3S,4S)-1-(benzenesulfonyl)-4-[methyl(pyrazin-2-ylmethyl)amino]pyrrolidin-3-ol