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1-[2-(1H-1,3-benzodiazol-6-yl)phenyl]ethan-1-one
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1-methyl-1H-pyrazole
(1R,5S)-8-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-3,8-diazabicyclo[3.2.1]octane
5-methoxy-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
(3aS,6aR)-5-(2,3-dihydro-1-benzofuran-5-carbonyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-(4-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-2-methyl-1,4-dihydropyridin-4-one
3-(1-butyl-1H-imidazol-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(3-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}propanamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
(1S,5R)-N-(2-fluorophenyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(oxan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
(1R,3s,6r,8S)-4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-4-azatricyclo[4.3.1.13,8]undecane
2-cyclopropyl-9-(3-methyl-2-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
(1-{3-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]propyl}piperidin-3-yl)methanol
(3R,4S)-1-[(4-fluorophenyl)methanesulfonyl]-4-propylpyrrolidin-3-amine
N-methyl-3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-ylmethyl}-1,2,4-oxadiazole-5-carboxamide
(3S,4S)-4-cyclopropyl-1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidine-3-carboxylic acid
[(2,6-difluoro-4-methoxyphenyl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-methoxy-2-methylpropanamide
(2S)-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(furan-3-carbonyl)pyrrolidine-2-carboxamide
7-methoxy-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyridin-3-ylmethyl)piperazine
1-(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-(pyrimidin-4-ylmethyl)piperidin-4-amine
(1R,5R)-N,N-dimethyl-6-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-methoxy-3-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-[(1R,5R)-6-[(3-phenoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N3-butyl-N5-cyclooctyl-N3-methyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
methyl 3-(furan-2-amido)-5-{[2-(2-methylphenyl)acetamido]methyl}benzoate
N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidin-4-amine
3-hydroxy-2-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
4-(2-methoxy-5-methylbenzenesulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-phenoxyethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
{2-[1-(1-benzofuran-5-ylmethyl)piperidin-2-yl]ethyl}dimethylamine
N-ethyl-5-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}pyrimidin-2-amine
[1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
6-{3-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
2-(3-fluoro-4-methoxyphenyl)-N-methylpyridine-4-carboxamide
3-[4-(morpholine-2-carbonyl)piperazin-1-yl]-1,2-benzothiazole
3-(2-methoxyethyl)-1-(2-methylphenyl)-5-(oxan-2-yl)-1H-1,2,4-triazole
1-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(1H-1,3-benzodiazol-1-yl)propan-1-one
ethyl({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-acetamidothiophene-2-carboxamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
3-(3-methoxyphenyl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1-ethyl-6-oxopiperidine-3-carboxamide