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5-methyl-2-(2-{4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}propyl)pyridine
N-[(2R)-oxolan-2-ylmethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[(cyclohexylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}piperidine-3-carboxylic acid
2-amino-6-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
(pentan-3-yl)[(2-phenoxypyridin-3-yl)methyl]amine
ethyl 4-({[1-(2-chloroprop-2-en-1-yl)-7-methyl-2-oxo-1,2-dihydroquinolin-3-yl]methyl}amino)piperidine-1-carboxylate
6-ethyl-2-(morpholin-4-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
N-(4-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
(5S)-4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,2,2,5-tetramethylpiperazine
ethyl 4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(methylsulfanyl)pyrimidine-5-carboxylate
4-methyl-6-[4-({[4-(methylsulfanyl)phenyl]methyl}amino)piperidin-1-yl]pyrimidin-2-amine
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)oxane-2-carboxamide
[1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methanamine
N-cyclohexyl-1-cyclopropyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1,2-oxazole-3-carboxamide
2-methyl-8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[2-(2,4-difluorophenyl)ethyl]-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidine
N-[(1-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperidin-3-yl)methyl]methanesulfonamide
2-methyl-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
2-[(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzonitrile
N-methyl-N-[2-(2-oxo-5,5-diphenylpiperidin-1-yl)ethyl]methanesulfonamide
4-(2-chloro-6-fluoro-3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
6-ethyl-4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-2-methylquinoline
3-{1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-acetamido-N-methylbenzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbut-3-enamide
N-(2,3-dimethylphenyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-({3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)benzoic acid
4-[1-(2-ethoxyacetyl)piperidine-4-carbonyl]-1-(4-methylphenyl)piperazin-2-one
5-(6-methoxynaphthalen-2-yl)-1H-1,2,4-triazole
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(4-fluoro-3-methylphenyl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
N-(2-methoxyethyl)-1-{1-[2-(3-methylphenyl)acetyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(4-hydroxyphenyl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-(methylamino)pyridine-4-carboxamide
1-(3-{[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenyl)ethan-1-one
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-[3-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
1-[1'-(pyridin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-methyl-3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
(1R,2R,3S,4S)-3-amino-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)bicyclo[2.2.1]heptane-2-carboxamide
2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1,3-benzothiazole
4-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(diethylamino)ethyl]-N-ethyl-5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(2S,4R)-4-(dimethylamino)-1-(isoquinolin-5-ylmethyl)pyrrolidine-2-carboxylic acid
2-[(4aR,7aS)-4-(2,5-dimethylfuran-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid