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5-ethyl-4-(pyrrolidin-1-ylmethyl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]furan-2-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-methyl-4-phenylthiophene-3-carboxamide
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-[(2R)-pyrrolidine-2-carbonyl]piperidine
5-[4-(2-methoxyethoxy)phenyl]-1-methyl-1H-indazole
2-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}pyridine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N4-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
4-(2,4-difluorobenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}furan-2-yl)methanol
7-(5-chloro-2-methoxybenzoyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(4-methyl-1H-pyrazol-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]propanamide
1-(furan-2-ylmethyl)-N-methyl-N-[3-(oxolan-2-yl)propyl]piperidine-4-carboxamide
(3S,4S)-4-cyclopropyl-1-(2,6-dimethylpyridine-4-carbonyl)pyrrolidine-3-carboxylic acid
3-{5-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-{[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]sulfonyl}benzonitrile
9-[2-(4-hydroxyphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(6-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-benzyl-4-[(3,5-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyridin-2-amine
6-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}pyridine-3-carbonitrile
N-(2-cycloheptylethyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-[(methylcarbamoyl)methyl]-3-oxo-N-(4-pentylphenyl)piperazine-1-carboxamide
2-{4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
N-(2-hydroxypropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(3-chlorobenzoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[2-(2-hydroxyethoxy)ethyl]urea
5-(2-chlorophenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}furan-2-carboxamide
4-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)benzoic acid
N-methyl-N-{[5-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)furan-2-yl]methyl}methanesulfonamide
2-{[4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-6-methylpyridine
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-{[(2-fluoroethyl)amino]methyl}-5,8-dimethylquinolin-4-ol
N-ethyl-6-(2-methoxyphenyl)-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 3-[(3S,4R)-1-[(4-hydroxy-3-methoxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
5-(3-chloro-2-fluorophenyl)pyridine-3-carboxamide
2-{2-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]-4-chlorophenoxy}acetic acid
3,3-diphenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
1-(6-fluoropyridin-3-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
1-[2-(dimethylamino)ethyl]-5-[4-(4-hydroxybutyl)piperazine-1-carbonyl]piperidin-2-one
5-benzyl-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(1-{[1-(pyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-2,6-dimethylquinoline
N-(oxan-4-yl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-(3,4-difluorophenyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-amine