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N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(1H-pyrazol-1-yl)acetamide
5-methyl-3-[(2R)-pyrrolidin-2-ylmethyl]-3,4-dihydroquinazolin-4-one
methyl 2-[1-(4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}phenyl)-N-methylformamido]acetate
5-({4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-N,N-dimethylfuran-2-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-2-(pyrrolidin-1-yl)benzamide
{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
1-(pentan-2-yl)-5-propyl-1H,4H-pyrazolo[3,4-d]imidazole
2-[ethyl({[(3R,4R)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
5-butyl-1-(3-methylphenyl)-4-(5-methylpyrazine-2-carbonyl)piperazin-2-one
(2S,4S)-4-amino-N-ethyl-1-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidine-2-carboxamide
4-chloro-5-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
4-[(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)methyl]morpholine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-(4-fluoro-2-methylbenzoyl)-2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}methanesulfonamide
5-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4-methyl-1H-imidazole
(1R,3S)-7-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-(2-hydroxyethyl)-6-[2-(propan-2-yloxy)propanoyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
3-ethyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridazin-3-amine
8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[3-(1H-indazol-1-yl)propyl]propanamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(phenylsulfanyl)ethan-1-one
3-(2-fluorophenyl)-3-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
(3S,5S)-1-[(4-hydroxy-3-methylphenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
6-{[cyclohexyl(methyl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
8-(1H-indol-2-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluoro-2-methoxyphenyl)-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}acetic acid
methyl[3-(methylsulfanyl)propyl](quinolin-2-ylmethyl)amine
2-{3-oxo-9-[2-(oxolan-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
5-methoxy-3-methyl-2-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indole
2-[(4-chlorophenyl)methyl]-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(furan-2-ylmethyl)piperidine-1-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-{2-oxo-2-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
(1R,5R)-3-benzoyl-6-[(2,3-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(2-butyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
(2S)-1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxylic acid
1-(2,6-dimethylpyridin-4-yl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazine
5-{[5-(oxan-2-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2R,3R)-3-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(4-benzylpiperazin-1-yl)-3-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]propan-1-one
3-(3-fluorophenyl)-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
(3R,5R)-1-benzyl-N-butyl-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-({3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide