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(1S,6R)-9-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-(6-hydroxy-6-methylheptan-2-yl)-3-(1,2-oxazinan-2-yl)propanamide
(1S,6R)-3-[(4Z)-hept-4-en-1-yl]-3,9-diazabicyclo[4.2.1]nonane
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-[3-(pyridin-3-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2R,3R,6R)-5-benzoyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-2-methoxy-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(furan-2-yl)-2-oxo-N-[3-(pyridin-2-yl)propyl]acetamide
N-[3-methoxy-4-(3-methylbutanamido)phenyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
(1R,2R,6S,7S)-4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
(1R,2R,6S,7S)-N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
2-hydroxy-5-[3-(1H-pyrazol-3-yl)phenyl]benzoic acid
1-[(4aR,8aS)-1-{[3-(benzyloxy)phenyl]methyl}-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-1H-indazole-3-carboxamide
5,6-dimethyl-N-[2-(pyridin-4-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
4-[1-(4-fluorophenyl)cyclopropanecarbonyl]-1-phenylpiperazine-2-carboxylic acid
2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}-2-(5-fluoro-2-methoxyphenyl)acetic acid
4-(4-fluoro-3-methoxyphenyl)-5-(3-methylbutyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-methyl-4-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]piperazin-2-one
(4aR,8aR)-7-[(2-cyclohexylpyrimidin-5-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-[3-(pyrrolidin-1-yl)phenyl]pyridine-3-carbonitrile
5-(2,3-dimethylphenyl)pyrazin-2-amine
[(1-benzylpyrrolidin-3-yl)methyl](methyl)[(1-methyl-1H-imidazol-5-yl)methyl]amine
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methoxy-3-methyl-1H-indole
(1S,5R)-6-[4-(difluoromethoxy)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
1-(3-phenylpropyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
1-[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-diphenylethan-1-one
5-[2-(4-chlorophenyl)-2-hydroxyacetyl]-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3,5-dimethyl-4-{6-methylimidazo[2,1-b][1,3]thiazole-3-amido}-1H-pyrazol-1-yl)acetic acid
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
2-cyclopentyl-N-{[(2S,4S)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}acetamide
9-(cyclohex-3-en-1-ylmethyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-hydroxyethyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(1S,5R)-3-[2-(2,3-difluorophenyl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(cyclopropylmethyl)-2-[(2S)-2-hydroxypropanoyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
7-fluoro-3-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]-1,2-dihydroquinolin-2-one
N-{4-fluoro-3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}propanamide
8-(furan-2-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
2-chloro-N-[1-(3-methylpyridin-2-yl)propyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-cycloheptyl-5-(2,3-dihydro-1H-isoindole-2-carbonyl)piperidin-2-one
2-(4-methyl-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidin-2-yl)phenol
8-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1,8-naphthyridine-2-carboxamide
ethyl 4-{10-oxo-3,9-diazaspiro[5.6]dodecan-3-yl}piperidine-1-carboxylate
2-(3,4-dimethoxyphenyl)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}acetamide
4-{1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine