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2-benzyl-9-[2-(methylamino)pyridine-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N,N-bis(prop-2-en-1-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[benzyl(methyl)amino]-3-[5-({[3-(dimethylamino)propyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[1-(2,4-dimethylphenyl)propyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-(2-chloro-4-fluorophenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(phenylsulfanyl)acetamide
(1S,5R)-1,3,3-trimethyl-6-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-6-azabicyclo[3.2.1]octane
[1-(3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propyl)piperidin-3-yl]methanol
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-5-(4-fluorophenyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
1-[(3-chlorophenyl)methyl]-4-(pyridin-4-yl)piperazine
5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
1-(furan-2-ylmethyl)-N-[2-(1H-imidazol-1-yl)ethyl]piperidine-3-carboxamide
N-methyl-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[2-(dimethylamino)-4-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-cycloheptyl-N-methyl-6-oxo-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
[4-(5-fluoro-4-methoxypyrimidin-2-yl)phenyl]methanol
5-(2-chloropyridine-4-carbonyl)-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(prop-2-en-1-yl)carbamoyl]piperidine-4-carboxylate
3-cyclohexyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-4-carboxamide
8-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(adamantan-2-ylmethyl)-6-{[(3-methoxypropyl)(1-methylpiperidin-4-yl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(2-methoxyethyl)-3-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
2-[(4-chlorophenyl)methyl]-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1'-[2-(4-fluorophenyl)-2-hydroxyacetyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
ethyl 2-{4-[(3-hydroxy-6-methylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxylate
1-[(5-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-2,4-dimethylphenyl)methyl]-4-methylpiperazine
ethyl 1-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-1-(4-methylphenyl)piperazin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(1H-pyrazol-1-yl)benzamide
3-{[6-(methoxymethyl)pyrimidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(1S,5R)-3-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-3,9-diazabicyclo[3.3.2]decan-10-one
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}furan-3-carboxamide
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-3-({3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
1-cyclopentyl-4-({[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine
7-chloro-4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]-2-methoxypyridine-3-carbonitrile
2-(2-{[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-[4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
(4-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-2,6-dimethylquinoline
3-(2,5-dioxopyrrolidin-1-yl)-N-[1-(4-methylpyridin-2-yl)propyl]benzamide
N-ethyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-methylpiperidine-1-sulfonamide