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5-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1,2-dihydropyridin-2-one
ethyl 1-{[3-({1-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-4-yl}oxy)phenyl]methyl}piperidine-2-carboxylate
5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N-ethylpyrimidin-2-amine
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
8-[2-(3-chloro-9H-carbazol-9-yl)acetyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
3,5-dimethyl-1-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-yl)-1H-pyrazole
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2-(propan-2-yl)pyrimidine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-2-yl)ethyl]amine
2-[5-(1-methanesulfonylpyrrolidin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
4-(4,4-difluoropiperidin-1-yl)-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
6-[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazine-1-carbonyl]-2-methylphenol
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1-methoxypropan-2-yl)piperidin-4-yl]propanamide
2-ethoxy-5-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}pyridine
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(3,4-dimethylbenzamido)pyrrolidin-1-yl]acetic acid
1-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-3-phenylpropan-1-ol
4-[5-(methanesulfonylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
4-[(3-methylthiophen-2-yl)sulfonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-(4-chloro-2-{[3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl}phenoxy)acetic acid
2-methyl-6-(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
5-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
8-(4-aminopiperidine-4-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[2-(trifluoromethyl)phenyl]methyl}-2-azaspiro[4.4]nonan-3-one
3-methyl-4-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
4-(5-chloro-2-methylbenzoyl)-1-phenylpiperazin-2-one
3,5-dimethyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1,2-oxazole-4-sulfonamide
2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]-N-(2-propyl-2H-1,2,3-triazol-4-yl)acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-acetamidoethyl)acetamide
4-phenyl-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-(2-hydroxyethyl)-8-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5S,8R)-N,N-dimethyl-3-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-3-azabicyclo[3.2.1]octan-8-amine
3-({4-[1-(thiophene-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2-methoxyethyl)(methyl)(2-{[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]oxy}hex-5-en-1-yl)amine
2-({1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
N-({5-[(2-chloro-6-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]pyridine-2,4-diol
3-{[(adamantan-2-yl)amino]methyl}-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-(3-methyl-1-oxo-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butan-2-yl)acetamide
(1R,5S)-3-(6-aminopyridine-2-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
(1R,3S)-3-methoxy-7-[4-(propan-2-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-acetamidopropanamide
4-(1H-imidazol-1-yl)-1-{[(4-methylphenyl)methyl]carbamoyl}piperidine-4-carboxylic acid
N-(2,1,3-benzothiadiazol-4-yl)-3-(pyrimidin-4-yl)piperidine-1-carboxamide
N-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]methanesulfonamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(4-{[(2S)-2-aminopropyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxy-2-methylpropan-1-one