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(1R,5R)-3-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3-azabicyclo[3.3.1]nonane
1-(4-methoxybenzoyl)-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperazine
4-{[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]methyl}-1,2-dihydrophthalazin-1-one
1-(1-{[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}cyclopentyl)-4-methylpiperazine
3-methyl-1-propyl-4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
(1H-imidazol-2-ylmethyl)({[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl})methylamine
methyl (1R,3S,3aR,6aS)-5-benzyl-1-ethyl-4,6-dioxo-3-(pyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
4-methoxy-N-[2-(methylsulfanyl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,6-dimethyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
3-(4-chlorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]urea
4-(2-methoxypyrimidine-5-carbonyl)-3,4-dihydro-2H-1,4-benzoxazine
2-(pyridin-3-ylmethyl)-9-(trimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-dimethyl-1H-indol-5-ol
3-ethyl-5-[3-(1H-imidazol-2-yl)phenyl]-1,2,4-oxadiazole
1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-4-methoxypiperidine
1-benzyl-N3-cyclopropyl-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-{2-[5-(2-chlorophenyl)furan-2-yl]-1H-imidazol-1-yl}-1-(pyridin-3-yl)ethan-1-ol
N-[2-(3-methoxyphenyl)phenyl]-1-(2-methylpropyl)piperidine-4-carboxamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
1-[3-methoxy-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole
1-(2-ethoxyphenyl)-4-[3-phenyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazine
2-(1-benzyl-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl)ethan-1-ol
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(trimethylpyrazin-2-yl)methyl]piperidin-4-ol
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-3-methylbutan-1-ol
5-acetyl-N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}thiophene-2-carboxamide
N-(4-chloronaphthalen-1-yl)-3-(methoxymethyl)pyrrolidine-1-carboxamide
7-[(5-methylfuran-2-yl)methyl]-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[(3S)-1-benzylpyrrolidin-3-yl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
7,7-dimethyl-2-[(pyrrolidine-1-sulfonyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N4-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-5,6-dimethylpyrimidine-2,4-diamine
2-(1-propylpiperidin-4-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
2-methoxy-4-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
4-(4-aminopyrimidin-2-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
2-{2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
N-butyl-2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamide
2-{4-[(3-hydroxypiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
4,6-dimethoxy-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-cyclopropyl-2-(1H-1,2,3,4-tetrazol-5-yl)-N-(thiophen-3-ylmethyl)benzamide
(3R)-1-{4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}pyrrolidin-3-ol
3-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}oxy)pyridine
1-ethyl-4-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazine
(1R,3S)-7-[(2-fluorophenyl)methyl]-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
2,4-dimethoxy-6-[4-(pyridin-2-ylmethyl)piperazin-1-yl]pyrimidine
1-cyclobutanecarbonyl-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
2-(azepan-1-yl)-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide