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N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1,1-dioxo-1λ6-thiolane-3-carboxamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]piperidin-4-amine
7-(cyclohexylmethyl)-2-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N3-benzyl-N5-[(2-chlorophenyl)methyl]-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-chloro-N-[2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
5-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1,3-oxazole-4-carboxamide
5-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]quinoxaline
N,N-dimethyl-1-(2-methylpropyl)-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-({4-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
methyl 4-({[(3S,5S)-1-(naphthalen-2-ylmethyl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
N-{2-methyl-1-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]propyl}acetamide
N-[(3-chlorophenyl)methyl]-3-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]propanamide
5-[2-(2,5-dioxo-1-propylimidazolidin-4-yl)acetyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-2-(methylamino)ethan-1-one
7-(cyclopropylmethyl)-2-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-({3-[(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)piperidine-2-carboxylate
5-methyl-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,3-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(naphthalen-2-yloxy)propanamide
2-(1-methyl-4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperazin-2-yl)ethan-1-ol
(2R)-2-amino-N-(1-cyclopentanecarbonylpiperidin-4-yl)-4-methylpentanamide
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
(3aR,6aR)-N,2-dimethyl-N-(quinoxalin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-tert-butyl-4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}furan-2-carboxamide
1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidine-4-carbonitrile
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(thiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(1H-indol-2-yl)phenyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
5-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-N-phenylpyrimidin-2-amine
5-oxo-1-(propan-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
[1-(2,5-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methanol
6-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-cyano-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-1H-pyrrole-2-carboxamide
5-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylpyrazine-2-carboxamide
3-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carbonyl)pyridine
5-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-{2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
10-methoxy-5-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2,6-diamino-4-[2-(dimethylamino)pyrimidin-5-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(4aR,7aS)-1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(dimethylamino)methyl]-1-[(1-ethyl-1H-indol-6-yl)methyl]pyrrolidin-3-ol
N-ethyl-4-{[4-(ethylamino)pyrimidin-2-yl]amino}piperidine-1-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-5-(1,2-oxazol-5-yl)furan-2-sulfonamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
1-[4-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-2-cyclopentylethan-1-one