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2-(3,4-dimethoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-(furan-2-yl)-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}azepane
2-(2,5-dioxoimidazolidin-4-yl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)acetamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
3-{[3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-3-oxopropyl](methyl)amino}-1λ6-thiolane-1,1-dione
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
N-(1-methyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
3-ethyl-5-hydroxy-N-[3-(4-hydroxyphenyl)propyl]adamantane-1-carboxamide
(3aR,6aR)-2-(carboxymethyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-methyl-1H-pyrrol-2-yl)-2-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]ethane-1,2-dione
5-{[4-(2-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
3-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}phenol
1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-(oxolan-3-yl)-1H-1,2,3-triazole
1-(4-methoxyphenyl)-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-one
1-benzyl-8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(3-ethoxyphenyl)-N-methylthiophene-2-carboxamide
N-cyclopropyl-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
1-benzyl-4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine
N-[(3-methylpyridin-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
3-({1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}methyl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(1H-pyrazol-1-yl)butan-1-one
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(1-propyl-1H-pyrazole-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-(2,4-dichlorophenoxy)ethan-1-one
1-{1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}piperidin-3-ol
N-[4-fluoro-3-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)phenyl]acetamide
2-methoxy-5-[(3-propoxypiperidin-1-yl)methyl]pyridine
ethyl 1-(2,3-dihydro-1H-inden-2-yl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine
(2R)-2-amino-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
7-{imidazo[1,2-a]pyridine-3-carbonyl}-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-fluoro-2-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
N-[2-(dimethylamino)ethyl]-5-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-fluoro-N-(3-{4-[2-(pyridin-2-yl)piperidin-1-yl]piperidin-1-yl}phenyl)benzene-1-sulfonamide
N-(2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
1-(cyclohexylmethyl)-N-(1H-imidazol-2-ylmethyl)piperidin-3-amine
6-[4-(3-methoxybenzoyl)piperazin-1-yl]-N,N-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(1S,5R)-6-benzyl-3-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5,7-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrido[2,3-d]pyrimidin-4-amine
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,6-dimethoxypyridine
N-(5-chloro-2-methoxyphenyl)-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-(1,3-thiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[1-(cyclohexylmethyl)-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-{[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-(1-{3-azaspiro[5.5]undecan-9-yl}piperidin-4-yl)-3-methylbutan-1-ol
1-[(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)methyl]azepane
N-{[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-[2-(naphthalen-1-yl)propan-2-yl]-3-(1H-pyrazol-4-yl)propanamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-6-(piperidin-3-yl)pyrimidin-4-amine