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4-methyl-2-propyl-6-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyrimidine
2-methoxy-5-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}pyrimidine
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methyl-1-(propan-2-yl)-1H-pyrazol-5-amine
N2,6-dimethyl-N4-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
1-{1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-3-yl}-1H-imidazole
N-(1-phenyl-1H-pyrazol-5-yl)-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(3,4,5-trimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
5-chloro-N-(2-oxopiperidin-3-yl)-3-phenyl-1H-indole-2-carboxamide
6-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
2-methoxy-N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-(thiophene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pyrrolidine-3-carboxamide
4-[(2-ethoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
2-[1-(3,4-difluorophenyl)-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(1-phenylpiperidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[2-(4-fluorophenyl)pyrrolidin-1-yl]propan-1-one
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
4-{[1-(2-methoxyphenyl)-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
N-(2-fluoro-4-methylphenyl)-3-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
N-(5-acetyl-2-ethoxyphenyl)-3-(dimethylamino)pyrrolidine-1-carboxamide
N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-2-(N-phenylmethanesulfonamido)propanamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(piperazine-1-sulfonyl)benzamide
N,3-dimethyl-1-propyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
5-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-(cyclopropanesulfonyl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(1H-imidazol-1-yl)ethyl]-N-methylpyridin-2-amine
2-({3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}methyl)pyrimidine
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
2-(3,4-dimethylphenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-amine
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methylpropyl)propanamide
1-[3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidine-3-carboxamide
4-amino-2-(1-benzofuran-2-yl)pyrimidine-5-carbonitrile
2-cyclohexyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1,3-benzoxazole-6-carboxamide
4-methyl-2-[1-(pyridin-4-yl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(4-fluorophenyl)-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
5-methoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}furan-2-carboxamide
8-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methoxy-4-[4-(piperidine-1-sulfonyl)phenyl]pyridine-3-carbonitrile
1-(3-fluorophenyl)-5-[(4-methyl-1H-pyrazol-1-yl)methyl]-1H-1,2,4-triazole
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
N-[1-(3,4-dimethylphenyl)propyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N,N-dimethyl-6-[3-(1H-pyrazol-1-yl)phenyl]pyrazin-2-amine