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({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
2-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
methyl 2-[(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}phenyl)formamido]acetate
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one
1-[(4-methylphenyl)methyl]-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazin-2-one
4-(1H-imidazol-1-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-ol
5-[4-(1H-pyrazol-3-yl)phenyl]-1,3,4-thiadiazol-2-amine
7-[(3,4-difluorophenyl)methyl]-2-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
4-[1,3-dimethyl-4-(4-phenyl-1H-imidazol-5-yl)-1H-pyrazol-5-yl]morpholine
N-[4-(oxolan-2-yl)butyl]piperidin-4-amine
3-(4-carbamoylphenyl)-5-hydroxybenzoic acid
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[2-(dimethylamino)ethyl]-N-{[7-fluoro-2-(2-methylphenyl)quinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
2-amino-4-(furan-3-yl)-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
4-methyl-1-[3-(2-methylphenyl)piperidin-1-yl]pentan-1-one
8-{[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]methyl}-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-2-one
5-acetyl-N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
(2S,4R)-N,N-diethyl-4-[5-(ethylsulfanyl)thiophene-2-amido]-1-methylpyrrolidine-2-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(quinoxalin-2-yl)-decahydro-1,6-naphthyridin-2-one
2-(methylamino)-N-(4-methylphenyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
3-[2-(2-phenylethyl)piperidine-1-carbonyl]pyridazine
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amino)ethan-1-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-(2-methoxy-5-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(pyrrolidin-3-yl)benzamide
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-sulfonamide
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
2-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
3-{[2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
1-{6-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}piperidine-4-carbonitrile
N-(3-hydroxypropyl)-2-methyl-N-(pyridin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-cyclohexyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
N-(2-methylbutyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-methoxyacetamide
S-[3-(4-cyanopiperidine-1-carbonyl)phenyl]-2,3-dihydroxy-N-methylpropane-1-sulfonamido
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-(3,5-difluorophenyl)-4-[(4-methylphenyl)methyl]morpholine-2-carboxamide
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
ethyl 1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxylate
N-{3-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
N-methyl-N-(2-phenyl-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
1-{5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
N-({2-[2-(hydroxymethyl)phenyl]phenyl}methyl)propanamide
1-(3-acetylphenyl)-3-[2-(ethylsulfanyl)ethyl]urea
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(3R,4S)-1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-methylthieno[2,3-d]pyrimidin-4-amine