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methyl 3-[1-(2-methanesulfonylacetyl)piperidin-2-yl]propanoate
6-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
5-(4-methoxyphenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2,4-triazin-3-amine
N-[3-(6-methyl-9H-purin-9-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
(2S)-1-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3-({3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)pyridine
3-(4-hydroxyphenyl)-N-(2-methanesulfonamidoethyl)-2-phenylpropanamide
3-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-1λ6-thiolane-1,1-dione
(3S,4S)-1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-[ethyl(pyridin-4-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
methyl 2-[(1-ethylpyrrolidin-3-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
N-(oxan-3-ylmethyl)-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
[3-(2-methoxyethyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
5-(hydroxymethyl)-2-methyl-4-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-3-ol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-[(cyclopropylmethyl)sulfanyl]acetamide
N-methyl-5-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2,4-oxadiazol-3-amine
8-(2-methoxypyridine-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-methyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
7-(5-chloro-2-methoxybenzoyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
3-[(2-fluorophenyl)methyl]-6-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-4H-thieno[3,2-b]pyrrole-5-carboxamide
(4aR,8aS)-6-(3-fluorobenzoyl)-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
4-{2,8-diazaspiro[4.5]decane-3-carbonyl}-1-(3-methoxyphenyl)piperazin-2-one
3-[(oxolan-3-ylmethyl)(propan-2-yl)amino]propanamide
N-[(2R,4R,6S)-2-(propan-2-yl)-6-[4-(1H-pyrazol-1-ylmethyl)phenyl]oxan-4-yl]acetamide
2-[4-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]ethan-1-ol
2-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]phenyl}-4-methyl-1,2-dihydrophthalazin-1-one
2-methoxy-1-{4-[3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-1-yl}ethan-1-one
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]hexan-1-ol
2-methyl-8-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(2,4-dimethoxy-3-methylphenyl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]furan-2-carboxamide
3-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
1-{1-[(1-hexylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(thiophene-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(4-methylphenoxy)piperidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
5-ethyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
3-methoxy-2,2-dimethyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
4-{1-[(2-methylphenyl)(pyridin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}benzoic acid
5-(3,4-dimethoxyphenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2,4-triazin-3-amine
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
methyl 6-[(4-hydroxy-3,5-dimethylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(5-phenyl-1,2,4-oxadiazol-3-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxylic acid