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5-(1H-indole-2-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]morpholine-2-carboxamide
5-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-cyano-N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}benzamide
N-(2,4-dimethoxyphenyl)-3-[1-(quinolin-2-ylmethyl)piperidin-4-yl]propanamide
(2S,4S)-4-[4-({[(2,5-difluorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-(1-{1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
3-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]propanoic acid
5-chloro-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(methylamino)benzamide
N-(6-methylpyridin-3-yl)spiro[2.5]octane-1-carboxamide
6-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]pyrimidin-4-ol
1-(1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}azetidin-3-yl)piperidine
methyl 2-[N-methyl-1-(6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)formamido]acetate
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
5-methyl-4-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-1-phenylpiperazin-2-one
3-(2-cyanophenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
1-{3-[(4-ethylpiperazin-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
3-{2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-4-ethylpiperazin-2-one
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N,N-dimethylazepan-4-amine
3-amino-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methoxypropan-1-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-[methyl(1H-pyrazol-3-ylmethyl)amino]-2-[3-(propan-2-yloxy)phenyl]acetic acid
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
(2S,4S,5R)-5-(3-chlorophenyl)-4-[(4-hydroxybutyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
(3aR,6aR)-2-[(3,4-dimethoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-chlorophenyl)methyl]-5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
1-(cyclopropylmethyl)-4-(4-methyl-1H-pyrrole-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
4-({[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl](methyl)amino}methyl)-1-tert-butylpyrrolidin-2-one
1-{1-[1-(1-benzothiophene-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-(pyrazin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)propanamide
N-(3-methoxyphenyl)-1-{2-[(2-methylphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
5-methoxy-2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-4H-pyran-4-one
(1H-indol-2-ylmethyl)({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]propanamide
3-hydroxy-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,2-oxazole-5-carboxamide
1-{4-[(2-methoxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-[1-(thiophen-2-yl)propyl]propanamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-3-(piperazin-1-yl)propan-1-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
4-benzyl-1-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
1-(4-benzoylpiperazin-1-yl)-4-(piperidin-1-yl)pentan-1-one
N-(2-chloro-6-methylphenyl)-3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidine-1-carboxamide
2-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-1,3-benzodiazole-4-carboxamide
2-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)azetidin-3-yl]pyridine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-(2H-indazol-2-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
2-methyl-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one