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N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylbutanamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decane
2-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)acetamide
N,5-dimethyl-N-(1-methylpiperidin-4-yl)-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-methoxyethyl)-1-(methoxymethyl)-N-(naphthalen-1-ylmethyl)cyclopropane-1-carboxamide
5-[(3-hydroxypiperidin-1-yl)methyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl]methanol
methyl 6-[(4-fluoro-3-methoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aS,8aR)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-(3-fluoro-4-hydroxyphenyl)-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]acetamide
3-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]pyridin-4-amine
4-[3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)pyridin-2-yl]morpholine
N-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-2-carboxamide
1-cyclopropyl-N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[2-(diethylamino)ethyl]-5-fluoroquinazolin-4-amine
1-(2-aminoethyl)-N-[2-(4-chlorobenzenesulfonamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1,4-dioxane-2-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(2-methoxyphenyl)propanamide
2-(2-ethylphenyl)-N-methylpyrimidin-4-amine
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(3-ethoxy-4-hydroxyphenyl)pyridine-3-carbonitrile
2-cyclopropyl-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
3-[4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]benzonitrile
(2S,4S)-N,N-diethyl-1-(4-fluorobenzoyl)-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
2-(2,3-dihydro-1H-inden-5-yloxy)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-methylpropan-1-one
5-cyclopropanecarbonyl-1'-(1-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-(azepan-1-yl)acetyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
2-(3,5-dimethyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)acetic acid
5-{2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
dimethyl(2-{2-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-ethyl-1-methyl-3-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-(2-methoxyethyl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-[2-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)ethyl]imidazolidin-2-one
N3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N5-cyclopentyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(1-cyclohexyl-1H-pyrazol-5-yl)acetamide
4-phenyl-5-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-imidazole
[3-(3-methoxypropyl)-1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]methanol
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-benzothiazole-6-carboxamide
(3aS,6aS)-2-cyclohexyl-5-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(2,4-dimethylbenzenesulfonamido)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-cyclohexanecarbonylpiperidine
6-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N-[(3-methoxyphenyl)methyl]-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
1-[(2-chlorophenyl)methyl]-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]azepan-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-6-fluoro-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide