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7-methoxy-3-[4-(pyrrolidin-1-ylmethyl)benzoyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
5-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-butyl-3-cyclopentyl-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazole
2-chloro-N-[1-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-butyl-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[(6-methoxy-2H-chromen-3-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
8-(3-aminopropanoyl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
[1-(5-chloro-2-methoxybenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
4-benzoyl-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propanoic acid
2-[3-(4-chlorophenyl)-5-[1-(2-oxopyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-(3-methoxypropyl)-9-(1,2,4-oxadiazol-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclohexyl-6-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,3-benzoxazole
methyl 3-{[2-(dimethylamino)ethyl]({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)carbamoyl}propanoate
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-methoxyphenyl)ethan-1-one
N-methyl-N-(pyrazin-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-{1-[4-(morpholine-4-carbonyl)pyridin-2-yl]piperidin-4-yl}-2-phenylethan-1-ol
1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-3-yl)propan-1-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperazine
5-[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
methyl (2S)-1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxylate
4-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)pyrimidin-2-amine
2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-2-methylpropanamide
2-methyl-3-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(naphthalen-1-ylmethyl)acetamide
6-methyl-2-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)pyridin-3-ol
N-(2-methoxyethyl)-1-[1-(2-methylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-5-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)-1,2,4-oxadiazole-3-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
(3S,4R)-1-(5-ethoxyfuran-2-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carboxylic acid
3-({[4-(pyridin-2-yl)butyl]amino}methyl)piperidin-3-ol
(3S,4R)-1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-4-methylpiperidine-3,4-diol
3,3-dimethyl-1-{2-oxo-2-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}urea
2-[(1S,5R)-6-[4-(4-methoxyphenyl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-hydroxyquinoxalin-2-yl)-N-methylpropanamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
1-(2-methanesulfonylethyl)-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazine
N4,N4-dimethyl-N6-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidine-4,6-diamine
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
ethyl 4-[(2S,4R,6S)-4-acetamido-6-(2-methylpropyl)oxan-2-yl]-1H-pyrazole-3-carboxylate
N,1-dimethyl-N-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
3-(1H-imidazol-1-yl)-N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]propanamide
2-{3-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenoxy}acetamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-methylpiperazin-2-one
1-{1-[6-(2-methoxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-[1-(2-methylpropanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide