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2-(1-methyl-1H-pyrazol-3-yl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-methyl-3-[(3S,4R)-3-(propan-2-yl)-4-[3-(thiophen-3-yl)propanamido]pyrrolidin-1-yl]propanamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine-3-carboxylate
2-cyclopropyl-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-hydroxypyrimidine-5-carboxamide
N-(3-cyclopentylpropyl)-4-methoxy-N-methyl-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
benzyl(methyl)({3-[3-(2-methylpropyl)morpholine-4-carbonyl]-1,2-oxazol-5-yl}methyl)amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(cyclopropylmethyl)-N-propyl-1H-pyrazole-3-carboxamide
3-methyl-4-oxo-N-[2-(propylsulfanyl)ethyl]-3,4-dihydroquinazoline-7-carboxamide
2-benzyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
N-[2-(pyridin-3-yloxy)propyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
7-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-8-fluoro-3,4-dihydroquinazolin-4-one
3-methyl-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-methoxy-3-methyl-N-(propan-2-yl)-1-benzofuran-2-carboxamide
1-benzyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
2-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-4-carboxamide
1-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-3-ol
N-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-N-methylpyrrolidine-3-carboxamide
1-{5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
methyl[1-(pyridin-3-yl)ethyl]{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
N3-[(2,6-difluorophenyl)methyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-1-benzofuran-5-carboxamide
2-(2-oxopiperidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1,5-dimethyl-4-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
{4-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)methyl]oxan-4-yl}methanol
1'-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-cyclopentyl-2-fluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-5-propyl-1,2-oxazole-3-carboxamide
(2S,4S)-4-amino-1-(1-carbamoylcyclopropanecarbonyl)-N,N-diethylpyrrolidine-2-carboxamide
4-(4-methoxy-2-methylphenyl)-6-methylpyrimidin-2-amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1H-1,3-benzodiazole-2-carboxamide
2-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}-4-(trifluoromethyl)pyrimidine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
2-amino-6-(2-fluoro-4-methoxyphenyl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
N-{4-[4-(4-formyl-1,4-diazepan-1-yl)piperidin-1-yl]phenyl}-2,4-dimethylbenzamide
7-methyl-2-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
2-(4-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}morpholin-3-yl)-N-(oxan-4-yl)acetamide
2-(3-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}phenyl)-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
3-fluoro-N-({7-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3-chloro-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-fluoro-N-methyl-1-benzothiophene-2-carboxamide
3-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylic acid
N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4-(piperidin-3-yl)benzamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
5-cyclobutyl-N-[3-(pyridin-3-yloxy)propyl]-1,3,4-oxadiazol-2-amine
3-(2-hydroxyphenyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide