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(1R,5S)-6-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(2R,3R)-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[1-(methoxymethyl)cyclopentyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(thiophene-2-sulfonamido)acetamide
(3R,4R)-4-cyclobutyl-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methylpiperidin-4-ol
N-methyl-N-[1-(pyridin-2-yl)propyl]piperidin-4-amine
2-(6-methoxypyridin-3-yl)-4,6-dimethylpyridine-3-carbonitrile
2-[6-(piperidin-1-yl)pyridin-3-yl]-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-[7-(6-ethylpyrimidin-4-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
5-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrazin-2-ol
N-methyl-N-(2-{methyl[(4-methyl-1H-imidazol-5-yl)methyl]amino}ethyl)cyclopentanamine
N-(1H-indol-4-ylmethyl)-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
5-(1,2-dihydroacenaphthylen-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-(thiophen-3-ylmethyl)-1,4-diazepan-6-ol
(2E)-3-(pyridin-4-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}prop-2-enamide
5-methyl-4-({[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
3-methanesulfonyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]benzamide
2-methyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,3-thiazole-4-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decane
9-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-5-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
1-(pyridin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperidine-4-carbonitrile
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][2-(3,4-dimethoxyphenyl)ethyl]methylamine
2-{4-[2-(2-methoxyphenoxy)acetyl]morpholin-3-yl}-N-methyl-N-propylacetamide
5-(4-fluoro-2-methoxyphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
4-(4-ethyl-1H-pyrazol-5-yl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine
9-ethyl-1-methyl-4-(oxan-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
2,6-dimethyl-4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]quinoline
1-cyclopentyl-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
3-(4-fluorophenoxy)-1-[(2,4,6-trimethoxyphenyl)methyl]azetidine
2-{2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
1-[4-(azonan-1-ylmethyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
8-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl 4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine-1-carboxylate
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3,5-dimethoxybenzamide
N-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}methanesulfonamide
1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
N-({5-[(3-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(thiophen-2-yl)ethyl]acetamide
5-(2-fluorophenoxymethyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-ethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
2-ethyl-5-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
(2S,4S)-4-{4-[4-(azepan-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
7-amino-4-[2-(cyclopentyloxy)phenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one