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ethyl 4-(7-chloro-3-{[N-cyclopropyl-1-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
N-[3-(furan-2-yl)phenyl]-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
N-[(3R,4R)-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-[4-(piperidin-1-ylmethyl)benzoyl]-2-(1,3-thiazol-2-yl)piperidine
4-(azonan-1-yl)pyrimidine-5-carboxylic acid
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)acetamide
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(5S,9aS,9bS)-2-phenyl-5-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(2-amino-2-methylpropanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2-{[4-(2,6-dimethoxypyridine-3-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
6-{[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]methyl}pyridine-2-carboxylic acid
7-[(4-fluorophenyl)methyl]-2-(3-methylbutyl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)hexan-1-one
(3aS,6aS)-2-[2-(2,3-dihydro-1H-indol-1-yl)acetyl]-5-pentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-hydroxypropanoyl)-N-(2-methoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
ethyl 2-({2-[3-(ethylcarbamoyl)pyrrolidine-1-carbonyl]phenyl}amino)acetate
4-(5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H-pyrazol-3-yl)phenol
1-{4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
5-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-(3-phenylpropyl)-1,3-benzoxazole
5-methyl-6-(4-methylpiperidine-1-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
4-[(3-fluorophenyl)methyl]-1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-1,4-diazepan-5-one
methyl 5-{[2-(2-hydroxyethoxy)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-(2,6-dimethylpyridin-4-yl)-4-(3-fluoropyridin-4-yl)piperazine
8-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxa-8-azaspiro[4.5]decane
4-methyl-N-{3-[methyl(phenyl)amino]propyl}-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[(4-methoxyphenyl)methyl]-5-(2-methylfuran-3-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4R)-1-{2-[(dimethylamino)methyl]benzoyl}-3,4-dimethylpyrrolidin-3-ol
4-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzoic acid
(2S)-2-amino-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(methylsulfanyl)butanamide
2-[4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)morpholin-3-yl]-N-phenylacetamide
methyl (2S)-2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}-3-(4-hydroxyphenyl)propanoate
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[1-(pyridin-4-yl)propan-2-yl]amine
2-{1-[2-(2-fluorophenyl)benzoyl]piperidin-3-yl}ethan-1-amine
2-methoxy-3-[1-(1-methylpiperidin-4-yl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridine
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-(3-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine-2-carbonitrile
8-[3-(pyridin-3-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-(1H-pyrrol-1-yl)butanamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
2-(dimethylamino)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-(3-methylphenyl)acetamide
2-amino-3-ethyl-N-[(4-ethylphenyl)methyl]-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,5-dihydro-1H-pyrrole
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-2,4,6-trimethylbenzamide
N-[(2R)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-1-oxobutan-2-yl]acetamide
2-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[5-(4-fluorophenyl)-6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl]acetamide
(2S,4R)-4-amino-N,N-diethyl-1-(3,3,3-trifluoropropanesulfonyl)pyrrolidine-2-carboxamide