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2-chloro-4-({methyl[2-(oxan-4-yl)ethyl]carbamoyl}amino)-N-propylbenzamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(4-methoxyphenyl)butan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(pyridin-4-ylsulfanyl)acetamide
4-(2,5-dimethoxyphenyl)-3-{[ethyl(methyl)amino]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[(2-hydroxyethyl)(methyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(thiophene-3-carbonyl)piperidine-3-carboxylate
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-cyclopentanecarbonylpiperidine-4-carboxamide
2-fluoro-6-[3-(1H-pyrazol-3-yl)phenyl]benzamide
2-amino-4-(6-methoxy-1H-indazol-3-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
4-(5-methylpyrimidin-4-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-1-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-{4-[(3-hydroxy-3-phenylpyrrolidin-1-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
1-phenyl-2-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}ethane-1,2-dione
N-[(2-fluorophenyl)methyl]-3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}propanamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-methoxy-4-methylbenzamide
2-(azepan-1-yl)-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-oxoacetamide
4-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}morpholine
2-[(1S,5R)-6-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-3-propyl-1H-pyrazole
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperidine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(3-methylthiophene-2-carbonyl)piperidine
4-(2-amino-5-methylpyrimidin-4-yl)-N,N-dimethylpiperazine-1-carboxamide
N-phenyl-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-methyl-2-[4-(trimethylpyrimidin-4-yl)phenyl]propanenitrile
2-(3-methylbutyl)-8-(2-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
2,6-diamino-4-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-phenyl-N-[(3R)-pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
N-(2-propyl-2H-1,2,3-triazol-4-yl)-2-(1H-1,2,3-triazol-1-yl)acetamide
1-(carboxymethyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-(4-aminoazepan-1-yl)-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
5-methyl-3-{3-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1,2,4-oxadiazole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(piperidine-1-carbonyl)pyridin-2-amine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
(4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}morpholin-3-yl)methanol
N-[(4-fluorophenyl)methyl]-2,2-dimethyl-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
N-(oxolan-2-ylmethyl)-1-(3-phenylpropyl)-N-propyl-1H-1,2,3-triazole-4-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(2-fluoro-4-methylphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(2,3,6-trimethylphenoxy)acetamide
2-({[(3R,4R)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-[2-(2-fluorophenyl)-1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-6-oxo-N-propyl-1,6-dihydropyridine-3-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](pyridin-4-ylmethyl)amine