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N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
(3R,5S)-N-[2-(dimethylamino)ethyl]-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidin-2-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-methoxy-5-methylphenyl)-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetic acid
8-(2,2-dimethylcyclopropanecarbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(furan-3-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2,6-dihydroxybenzamide
N,N-dimethyl-4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazine-1-carboxamide
N-(4-chloro-3-methylphenyl)-2-[(3-hydroxyadamantan-1-yl)amino]acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylacetamide
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)urea
1-(4-ethylpiperazin-1-yl)-3-[1-(6-methoxypyridine-3-carbonyl)piperidin-4-yl]propan-1-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(azepane-1-carbonyl)-N-benzyl-N-methyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[4-(3-chlorophenyl)-5-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
6-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)pyridine-2-carboxylic acid
(2S)-2-amino-N-[1-benzyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-cyclopropylacetamide
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[4-(1H-pyrazol-1-yl)phenyl]methyl})amine
1-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-cyclohexyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
4-{[1-(1,1-dioxo-1λ6-thiane-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
4-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4H-chromene-3-carboxamide
6-ethyl-2-methyl-4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]quinoline
2-{2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
N-cyclopropyl-5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(1S,5R)-6-[(1-ethyl-1H-indol-6-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2-{2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]-6-methoxyphenoxy}ethyl)dimethylamine
2-[(4-chlorophenyl)methyl]-8-(2-hydroxybutyl)-2,8-diazaspiro[4.5]decan-3-one
methyl N-{1-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-1-oxopropan-2-yl}carbamate
3-{[1-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
4-[2-(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-2-yl)ethyl]morpholine
4-[5-(oxan-4-ylmethyl)-1,2,4-oxadiazol-3-yl]-1H-indole
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
4-(3-chloropyridin-4-yl)-3-methyl-1-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperidin-3-ol
3-(2-methoxyethyl)-1-{[(4-methoxyphenyl)methyl]carbamoyl}piperidine-3-carboxylic acid
9-(oxane-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(dimethylamino)-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)benzamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(furan-2-yl)propanamide
1-{2-[1-(5-chloro-3-methyl-1H-indole-2-carbonyl)piperidin-2-yl]ethyl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
4-(3-phenylpropyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-[(2S)-oxolan-2-ylmethyl]-4-pentyl-1H-1,2,3-triazole
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-(3-hydroxyphenyl)-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyrrolidin-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(thiophen-2-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione