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N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-methyl-2-(morpholin-4-yl)-N-[2-(pyrazin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
3-(2-fluorophenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-(2-{methyl[(5-propylfuran-2-yl)methyl]amino}ethyl)piperidin-2-one
1-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
3-(4-methyl-1,3-thiazol-5-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
4-{2,2-dimethyl-3-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propyl}morpholine
2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(cyclohexylmethyl)-5-[(2-methoxyethyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-2,4-dioxo-N-(2-phenoxyethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[4-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decane
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
{3-[(2-fluorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-3-yl}methanol
N-(3-methoxypropyl)-4-[(pyridin-4-ylmethyl)sulfamoyl]benzamide
2-methoxy-3-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}quinoline
2-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-(3-methylphenyl)-5-{1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-2-yl}pyrimidine
1-(4-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
2-{3-[4-(1,3,5-triazin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl][(1-phenylpyrrolidin-3-yl)methyl]amine
2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
methyl 3-({[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}amino)benzoate
1-(oxolan-3-ylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
methyl 2-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}piperidine-1-carboxylate
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2,6-dimethoxypyrimidine
[1-({[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)amino}methyl)cyclopentyl]methanol
(2S)-2-amino-1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-3-(1H-imidazol-4-yl)propan-1-one
2-amino-6-cyclobutyl-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(cyclopropylmethyl)-3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}-1-(pyridin-3-yl)ethan-1-ol
1-(cyclobutylmethyl)-3-({[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
4-ethyl-1-[(3-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one
3-chloro-N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-4-methylbenzamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-propyl-1,2-oxazole-4-carboxamide
1-(3-methyl-1H-pyrazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}oxane-4-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(3R,4S)-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-4-propylpyrrolidin-3-amine
1-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidin-3-yl)-2-methylpiperidine
2-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethan-1-ol
2-({[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
8-methyl-5-(2-methyl-1H-imidazol-4-yl)quinoline
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
3-cyclopropyl-1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide
8-{2-[ethyl(methyl)amino]acetyl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{2-[4-(methylsulfanyl)phenyl]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
6-amino-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyridine-3-carboxamide