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[(5-chloro-2,3-dimethoxyphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-methyl-4-{4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]phenyl}piperazine
2-(2,6-dimethylpyrimidine-4-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
(2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-yl)methanol
1-(2-chlorophenyl)-4-{[3-(difluoromethoxy)phenyl]methyl}piperazin-2-one
(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-(5-methylpyrazine-2-carbonyl)-8-azabicyclo[3.2.1]octane
[(2S,6S)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(1,3-thiazol-2-yl)piperidin-4-ol
6-(4-phenyl-1,4-diazepane-1-carbonyl)-1,2,3,4-tetrahydroquinoxaline-2,3-dione
[2-oxo-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethyl]urea
N-(cyclobutylmethyl)-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)-N-(oxolan-2-ylmethyl)acetamide
1-(3-hydroxypropyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
1-(adamantan-1-yl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazine
(1S,5R)-6-(cyclobutylmethyl)-3-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
5-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-(4-oxo-4-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}butyl)pyrrolidin-2-one
{4-[(2-chlorophenyl)methyl]-1-[3-(methylsulfanyl)propyl]piperidin-4-yl}methanol
N-[(4-methoxyphenyl)methyl]-5,6-dimethyl-N-(2-methylpropyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)benzamide
(3R,4S)-4-phenyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-amine
1-[1-(adamantan-2-yl)piperidin-3-yl]-4-phenylpiperazine
N-{[1-(furan-3-ylmethyl)piperidin-3-yl]methyl}-4-phenylbenzamide
1-(3-methylpyridin-2-yl)-4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazine
5-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridine-2-carbonitrile
4-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-dimethylpiperazine
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
(3R,4R)-4-(morpholin-4-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-sulfamoylbenzamide
4-{2-[1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}phenol
N-methyl-3-(morpholine-4-carbonyl)-1-propyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]propane-1,2-diol
methyl (2S,4S,5R)-5-(4-chlorophenyl)-4-[(2-methoxy-2-oxoethyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
4-[(4-methyl-1H-imidazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]({[5-(2-fluorophenyl)furan-2-yl]methyl})methylamine
3-{[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(4-hydroxyphenyl)methyl]-4-[(1S)-1-phenylethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1,3,4-thiadiazole
N-(carbamoylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-({1-[4-(1H-pyrazol-5-yl)benzoyl]piperidin-4-yl}oxy)pyridine
N-[2-(pyridin-2-ylsulfanyl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2,6-dimethylquinoline-4-carboxamide
4-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)morpholine
(4S,4aS,8aS)-1-(2,6-difluorobenzoyl)-4-phenyl-decahydroquinolin-4-ol
2-({[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino}methyl)-6-methylquinolin-4-ol
N-[(2-methylphenyl)methyl]-2-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
[(2S,6S)-4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-[2-(4-methoxyphenyl)ethyl]-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide