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1-methyl-4-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}piperazine-2-carboxylic acid
4-(1-{1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-4-yl}ethyl)morpholine
6-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,4R)-4-(4-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl]acetamide
(2S,4R)-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-(4-{2-[4-(3-methylpyridin-4-yl)piperazin-1-yl]acetamido}phenyl)acetamide
4-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(2-methoxyphenyl)propan-1-one
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
1-(3-{[3-(3-hydroxypiperidine-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
3-(methylsulfanyl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
1-{3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
6-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]quinoxaline
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)acetamide
5-methyl-3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}-1,2-oxazole
6-ethyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
3-methyl-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1-[2-(trifluoromethoxy)phenyl]urea
2-(carbamoylamino)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}acetamide
1-[1-(4-chlorobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-{[(cyclobutylmethyl)(oxolan-2-ylmethyl)carbamoyl]amino}-4-methoxybenzoate
N-({7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methoxy-2-phenylacetamide
5-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
1,9-dimethyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-3-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N3-cyclohexyl-1-cyclopropyl-4-oxo-N5-[2-(4-phenylpiperidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamide
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
N-methyl-N-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}oxolan-3-amine
3-cyclopentyl-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-phenyl-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl][2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amine
4-chloro-2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indole
3-{5-[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-1,2,3-triazol-4-yl]thiophen-3-yl}prop-2-yn-1-ol
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-[(3S,4R)-1-[3-(3,4-dimethylphenyl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
3-{[(2-hydroxyphenyl)methyl]amino}-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
3-(5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylazepane-2-carboxamide
3-(2-fluoro-5-methoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2-(3-methoxyphenyl)pyrrolidine
1-(3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-7-methylimidazo[1,2-a]pyridine-2-carbonyl)azepane
(4aR,6R,8aS)-2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-(3,4-dimethoxyphenyl)-1-benzofuran-2-carboxamide