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(3S,4R)-1-(2-aminopyridine-4-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
7-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
3-methoxy-1-{2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
5-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropyl}morpholine
1-[1-ethyl-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-[2-(1H-imidazol-4-yl)ethyl]-5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-(1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)propan-1-one
5-(dimethylamino)-2-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
N-cyclooctyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-[4-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)-1H-pyrazol-1-yl]propanoic acid
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]propanamide
5-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-2-phenylpyrimidin-4-ol
1-(1-cycloheptylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
2-[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]ethan-1-ol
1-[(5-methylpyrazin-2-yl)methyl]-5,5-diphenylpiperidin-2-one
2-[({1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
5-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1,3-dimethyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazole-5-carboxamide
3-({[3-(4-chloro-1H-pyrazol-1-yl)propyl]amino}methyl)piperidin-3-ol
N-({7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3-(1-methyl-1H-pyrrol-2-yl)-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
6-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-N-(propan-2-yl)pyridazin-3-amine
1-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]ethan-1-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
2-{2-[1-(4-chloro-2-hydroxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
[(2-methoxyphenyl)methyl](oxolan-3-ylmethyl)(pyridin-3-ylmethyl)amine
N-methyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
methyl (2S,4R)-1-[(3-fluorophenyl)methyl]-4-(3-methoxybenzamido)pyrrolidine-2-carboxylate
(1S,4R)-2-[2-(benzenesulfonyl)ethyl]-2-azabicyclo[2.2.1]heptan-3-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2,5-dimethylphenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1,3-diazinane-2,4-dione
3-[({5-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]furan-2-yl}methyl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{[(3R,4R)-1-(3,4-dimethoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
3-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
(3S,4R)-3-benzyl-4-methyl-1-(1-phenylcyclopropanecarbonyl)piperidin-4-ol
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-2-one
4-{2-[(4aR,8aS)-6-(2-fluorobenzoyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-7-methyl-2H-chromen-2-one
N-[(3S,4R)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(1H-indol-4-ylmethyl)-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
8-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-3-oxopropyl]imidazolidine-2,4-dione
4-{[1-(2-fluorophenyl)-1H-pyrrol-2-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(3R,4R)-4-(hydroxymethyl)-1-[(5-propylfuran-2-yl)methyl]piperidin-3-ol
(2-{2-[1-(4-fluoro-3-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide