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5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(4-methoxypiperidin-1-yl)sulfonyl]pyrrolidin-3-yl]methanol
4-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
(3aR,6aR)-2-[(5-chlorothiophen-2-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(5-methoxy-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
3-{[(3R,4S)-3-amino-4-(2-hydroxyethyl)pyrrolidin-1-yl]sulfonyl}-N-phenylbenzamide
5-methoxy-6-(4H-1,2,4-triazol-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
2-cyclopropyl-N-[3-hydroxy-1-(4-methylphenyl)propyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-[(4-methoxyphenyl)methyl]-8-methyl-4-oxo-N-propyl-1,4-dihydroquinoline-3-carboxamide
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-3,5-dimethyl-1H-pyrazole-4-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-phenoxyethyl)piperazine
2-[(1S,5R)-6-[(1-ethyl-1H-indol-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
1-(4-methoxy-2-methylphenyl)-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
1-(2-chlorophenyl)-3-{1-[1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-benzyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
(1R,5R)-N,N-dimethyl-6-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(5-chloro-1H-indol-2-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-phenoxypropan-1-one
2-(5-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-3-yl)acetamide
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
methyl 6-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}carbamoyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
7-(propan-2-yl)-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-(2,4-difluorophenyl)ethyl]-1-(1H-pyrazole-4-carbonyl)piperidine
3-(3-fluoro-4-phenylbenzoyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
N-methyl-3-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}benzamide
2-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
(1R,5S,8S)-N-[4-(furan-2-yl)phenyl]-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
4-(3-chloro-2-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
methyl 3-{4-phenyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}propanoate
2,4-dimethyl-6-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyrimidine
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
3-[(benzylamino)methyl]-6,7-dimethoxy-1-[(4-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
N,N-dimethyl-4-[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carbonyl]piperazine-1-carboxamide
1-methyl-N-propyl-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}butanoic acid
2-[2-(butan-2-yl)phenoxy]-1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}ethan-1-one
3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]propan-1-ol
4-[4-(6-methoxypyridin-2-yl)benzenesulfonyl]morpholine
3-({[(1-ethyl-1H-imidazol-5-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
methyl 3-(1-methyl-1H-imidazol-2-yl)benzoate
N,3-dimethyl-1-propyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one