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2-(dimethylamino)-2-(3-methylphenyl)-N-[3-(pyridin-2-yl)propyl]acetamide
1-[3-(methylsulfamoyl)phenyl]-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
3-(2-methylphenyl)-1-[4-(pyridin-3-yl)pyrimidin-2-yl]pyrrolidin-3-ol
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
4-benzyl-1-[2-(thiophen-3-yl)acetyl]-1,4-diazepan-5-one
(3aS,6aS)-2-[(2-ethylpyrimidin-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(6-chloropyridin-3-yl)methyl](2-methoxyethyl)(thiophen-2-ylmethyl)amine
4-{4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}thiomorpholine
N-(2-methoxyethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
4-(3-fluorophenoxy)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylic acid
1,3-dimethyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(oxolan-3-yl)acetamide
[2-({1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}oxy)ethyl]dimethylamine
6-[(2-hydroxyethyl)(methyl)amino]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-[(3R,4S)-4-(5-methylfuran-2-yl)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]pyrrolidin-3-yl]methanesulfonamide
N-ethyl-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)furan-3-carboxamide
1'-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-butyl-4-methyl-6-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]pyrimidin-2-amine
N-[1-(4-fluorophenyl)-2-hydroxyethyl]quinoxaline-5-carboxamide
6-[3-(1-methoxyethyl)phenyl]-N,N-dimethylpyrazine-2-carboxamide
N4-[1-(4-fluorophenyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
[(2-cyclohexylpyrimidin-5-yl)methyl](isoquinolin-5-ylmethyl)methylamine
2-{1-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propyl]pyrrolidin-2-yl}-1,3-thiazole
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[(3-methylquinoxalin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(2S,4S)-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}urea
4-[2-(3,4-dimethoxyphenyl)ethyl]-4H-1,2,4-triazole
N-(1-benzylpiperidin-4-yl)-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
N-[(2S)-2-aminopropyl]-4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzamide
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(carbamoylmethyl)acetamide
N-({5-[(1-ethyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
3-{[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
methyl 3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-5-(cyclobutylmethoxy)benzoate
3-methyl-1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
8-(2-hydroxyethyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-3-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
5-butyl-1'-(2-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-{[1-(pyridin-3-yl)propan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N'-cyclopentyl-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)butanediamide
1-(4-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]sulfonyl}phenyl)ethan-1-one
N-(dicyclopropylmethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-N-[(4-methylphenyl)methyl]quinazolin-4-amine
N-({5-[(2,4,5-trimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclopropanecarboxamide
2-(4-methanesulfonylphenyl)-1-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-imidazole
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-phenyl-1,2-dihydropyridin-2-one
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide