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9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(1-cyclohexyl-5-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-6-yl}-1H-1,2,4-triazol-3-yl)acetamide
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
6-amino-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]hexan-1-one
3-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-2H-chromen-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-(2-methoxy-5-methylphenyl)-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
8-methoxy-5-(1-methyl-1H-imidazol-2-yl)quinoline
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(propan-2-yl)pyrimidin-2-amine
3-{2-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}-1λ6-thiolane-1,1-dione
N-{1-[(1-propyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-1H-pyrazol-5-yl}pyridine-4-carboxamide
1-[1-(2-phenylethyl)-5-[2-(thiophen-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
(2R,3R,6R)-5-(3,6-dimethylpyrazin-2-yl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
14-(3,4-dihydroxyphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{[2-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]amino}acetic acid
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-(3,4-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4S)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(2-propyl-2H-1,2,3-triazol-4-yl)-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
1-ethyl-5-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
8-[5-(methoxymethyl)furan-2-carbonyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
1-[(4aR,8aS)-6-(5-acetylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-cyclohexylpropan-1-one
5-(azocane-1-carbonyl)-1-cyclopropylpiperidin-2-one
N-(1-benzylpiperidin-4-yl)-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(methylamino)pyrimidine-5-carboxamide
2-[2-(furan-2-yl)-1H-imidazol-1-yl]-5-methylphenol
(5S,9aS,9bS)-5-(2-fluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-ethyl-1-[3-(1H-imidazol-5-yl)phenyl]-3-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]urea
4-{1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-methylpropan-2-yl}morpholine
1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-{1-[3-(1H-indazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}benzonitrile
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
(3S,5R)-5-(morpholine-4-carbonyl)-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-propylbenzoyl)piperidin-3-yl]propanoic acid
3-{[3-(3-chlorobenzoyl)piperidin-1-yl]sulfonyl}pyridine
methyl 4-(1H-1,3-benzodiazol-1-yl)-1H-pyrrole-2-carboxylate
2-[4-(4-acetylphenyl)piperazin-1-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(4-methylthiophen-2-yl)pyridine-3-carboxamide
3-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]urea
[4-({4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
N-{1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-yl}-N-methylacetamide
methyl (1R,3S,3aR,6aS)-3-(2-chloro-4-hydroxyphenyl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
methyl 2-hydroxy-5-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}methyl)benzoate
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
(2S)-2-hydroxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-phenylpropan-1-one
4-hydroxy-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidine-4-carboxylic acid
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-3-(1H-pyrazol-4-yl)propanamide
1-[1'-(5-hydroxypyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one