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N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]cyclobutanecarboxamide
6-(isoquinolin-5-yl)pyrazine-2-carboxamide
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
{4-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]morpholin-3-yl}methanol
2-(butan-2-ylsulfanyl)-5-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}pyrimidine
1-({1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
(2S,4S)-1-benzyl-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
3-methyl-3-phenyl-1-(1H-pyrazole-4-sulfonyl)piperidine
methyl 3-[(2,3-dihydro-1-benzofuran-2-ylformamido)methyl]-5-[3-(trifluoromethyl)benzamido]benzoate
2-{3-[1-(but-2-yn-1-yl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-[(4-methoxyphenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-chloro-N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
5-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}pyrimidin-2-amine
6-methyl-3-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(ethoxymethyl)-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine
3-(morpholine-4-carbonyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-{1-[(methylcarbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
N-(2-methoxyphenyl)-3-(2-phenylacetyl)piperidine-1-carboxamide
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-[4-(propan-2-yloxy)phenyl]acetic acid
(2E)-3-(2-chlorophenyl)-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylprop-2-enamide
(furan-3-ylmethyl)({[3-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl})methylamine
1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-methanesulfonyl-1,4-diazepane
4-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(pyridin-4-yl)acetamide
1-(carbamoylmethyl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
2-oxo-1-(2-propoxyethyl)-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[1-(cyclohexylcarbamoyl)piperidin-4-yl]-2-(ethylamino)pyrimidine-5-carboxamide
2-(4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
2-acetamido-N-[(2-methoxyphenyl)methyl]-3-methyl-N-(prop-2-en-1-yl)butanamide
({3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
2-tert-butyl-6-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)phenol
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]quinoline
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
(3S,4S)-4-(piperidin-1-yl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-ol
N-[3-(dimethylamino)propyl]-4-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
1-(cyclohexylmethyl)-5-[(1-hydroxy-2-methylpropan-2-yl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-methoxy-2-methylphenyl)-2-[4-(morpholine-4-carbonyl)piperidin-1-yl]acetic acid
2-[(3-benzoylpiperidin-1-yl)methyl]pyridine-3-carboxylic acid
1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
[1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-N-methyl-N-(propan-2-yl)propanamide
(3R,4S)-4-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(ethyl)amino]oxolan-3-ol
methyl({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl})[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
5-chloro-3-[1-(1H-imidazol-1-yl)butan-2-yl]-3,4-dihydroquinazolin-4-one