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1-cyclopentyl-4-(2-methylfuran-3-carbonyl)-1,4-diazepan-6-ol
4-{2,2-dimethyl-3-[3-(2-methylphenoxy)azetidin-1-yl]propyl}morpholine
2-[4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperazin-1-yl]pyrimidine
N-[(2S,4R,6S)-2-(4-methyl-1H-imidazol-5-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
N2-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
(7S,9aR)-6,9-dioxo-N-phenyl-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
12-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
methyl 2-(azepane-1-sulfonyl)-6-benzyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl[2-(2-methyl-1H-indol-1-yl)ethyl]{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
3-{5-[(3-methyl-3-phenylpiperidin-1-yl)methyl]-1,3,4-oxadiazol-2-yl}pyridine
5-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
4,6-dimethyl-2-oxo-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(3-hydroxyphenyl)-2-[methyl(thiophen-2-ylmethyl)amino]acetic acid
[(3R,4R)-4-[(dimethylamino)methyl]-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-3-yl]methanol
2-(1H-1,3-benzodiazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
ethyl 2-{1-azabicyclo[3.2.1]octan-5-yloxy}benzoate
N,N-dimethyl-5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-amine
N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(3S,4S)-4-(propan-2-yloxy)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-ol
1-[(1R,5R)-6-[(6-methoxynaphthalen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(4-chlorobenzoyl)piperidine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}propyl)pyrrolidin-2-one
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}but-3-en-1-one
2-[2-(morpholin-4-ylmethyl)phenyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(4-methoxybenzoyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
(3S,4S)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-propylpyrrolidine-3-carboxylic acid
(1-benzofuran-2-ylmethyl)(methyl)[3-(1-methyl-1H-pyrazol-4-yl)propyl]amine
5-methyl-2-(3-methylthiophen-2-yl)-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
(4aS,7aR)-1-(2-methyl-4-phenylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-{1-benzyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-4-chloro-1-methyl-1H-pyrazole
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-[4-(dimethylamino)azepan-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(ethylamino)-N-[3-methoxy-4-(3-methylbutanamido)phenyl]-4-methyl-1,3-thiazole-5-carboxamide
N-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)benzamide
3-[2-amino-4-methyl-6-({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amino)pyrimidin-5-yl]propanoic acid
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methylthiophene-2-carboxamide
(3R,4S)-3,4-dimethyl-1-(1,3-thiazol-2-ylmethyl)piperidin-4-ol
S-(4-fluoro-3-methylphenyl)-2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethane-1-sulfonamido
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-amine
N-{4-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]phenyl}acetamide