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1-{5-[(3-chlorophenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl}butan-2-ol
(3aR,5R,6S,7aS)-N-(4-hexylphenyl)-5,6-dihydroxy-octahydro-1H-isoindole-2-carboxamide
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-sulfonyl]-N-(2-ethoxyethyl)benzamide
3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}urea
(3R,4R)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
8-{[4-(difluoromethoxy)phenyl]methyl}-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
2-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenol
(3R)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
1-(2-benzylmorpholin-4-yl)-3-(3,4-dimethyl-1H-pyrazol-5-yl)propan-1-one
(3aS,6aS)-2-(ethanesulfonyl)-5-[(3-fluoro-2-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3-methoxypiperidin-4-amine
3-[(1-ethyl-1H-imidazol-2-yl)methyl]-7,8-dimethyl-3,4-dihydroquinazolin-4-one
1-{[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
5-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2S,4R)-1-(3-chloro-4-hydroxybenzoyl)-4-cyclopropaneamido-N-ethylpyrrolidine-2-carboxamide
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-5-[(pyridin-2-ylformamido)methyl]benzoate
1-cyclobutanecarbonyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(1H-imidazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[2-({[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
2-(4-fluorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)acetamide
4-{2-[4-(methylsulfanyl)phenyl]ethyl}-1λ6-thiomorpholine-1,1-dione
(1S,5R)-3-cyclobutanecarbonyl-N-(3-methoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-fluorophenoxymethyl)piperidine
(3aR,7aS)-N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
4-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-1-phenylpiperazin-2-one
2-(4-acetylpiperazin-1-yl)-N,N-bis(prop-2-en-1-yl)acetamide
(4aR,7aS)-1-acetyl-4-[(2-methoxy-3,5-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
8-chloro-2-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}quinolin-4-ol
1-(2-methoxyphenyl)-4-(4-phenylbutanoyl)piperazin-2-one
3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl({2-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]ethyl})amine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-phenylacetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
3-ethyl-4-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
(1S,4S)-2-(3-chlorophenyl)-5-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
1-{1-benzyl-5-[3-(5-methylfuran-2-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
5-[4-(morpholin-4-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1,3-dimethyl-2,6-dioxo-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-benzyl-4-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperazin-2-one
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
2-methoxy-N-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide