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1-[2-(dimethylamino)ethyl]-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
methyl 1-[methyl({[2-(trifluoromethyl)phenyl]methyl})carbamoyl]cyclopropane-1-carboxylate
5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
6-tert-butyl-3-(1H-imidazol-2-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-chloro-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
N-(6-methoxypyridin-3-yl)-3-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
2-(adamantan-1-yl)-N-ethyl-4-hydroxy-N-(2-hydroxyethyl)pyrimidine-5-carboxamide
N-{[3-(difluoromethoxy)phenyl]methyl}-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[3-(benzyloxy)azetidine-1-carbonyl]piperidin-1-yl}propan-1-one
2-(dimethylamino)-8-(3-phenoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}-1λ6-thiane-1,1-dione
1-(5-methylhex-5-en-2-yl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
2,3,5,6-tetramethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
(3S,4R)-N-(2-chlorophenyl)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carboxamide
3-methyl-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]butan-1-one
ethyl 2-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-2-yl}acetate
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-methyl-2-(pyridin-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
1-{4-[3-(3-methylphenoxy)azetidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-[(3R,4R)-1-[2-(1,2-benzoxazol-3-yl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamide
2-(2-methyl-1H-imidazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
1,3-dimethyl-2,6-dioxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-propyl-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyrrolidin-2-one
8-(2-hydroxyacetyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
3-{4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[2-(3-hydroxyphenyl)acetyl]pyrrolidine-2-carboxamide
2-[3-(oxolan-3-yl)-5-(piperidin-4-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-pentanamidobenzamide
2-(quinolin-2-ylmethyl)-1,2-dihydrophthalazin-1-one
2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-N-(propan-2-yl)pyridine-4-carboxamide
3-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1-(2-fluoropyridin-3-yl)urea
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(piperazine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
2-(2-hydroxyethyl)-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[(5-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
N-[(3,4-difluorophenyl)methyl]-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
4-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-[(3,4-difluorophenyl)methyl]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
(3aR,6aR)-2-{[6-(dimethylamino)pyridin-3-yl]methyl}-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 2-(1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperidin-2-yl)acetate
4-[2-(2-methoxy-4-methylphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-3-phenoxybenzamide
N-methyl-2-[3-oxo-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazin-2-yl]acetamide
2-(4-chlorophenyl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 4-{1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}piperazine-1-carboxylate