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1-{3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenyl}ethan-1-one
4-[({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amino]-2-methoxypyridine-3-carbonitrile
N-[3-(methylsulfanyl)propyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
3-(2-hydroxyphenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
2-(4,5-dimethyl-1H-imidazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(1-methylpiperidin-4-yl)methyl]-2-phenylacetamide
N-cyclohexyl-3-({[(4-fluoro-3-methoxyphenyl)methyl]amino}methyl)-N-methylpyridin-2-amine
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(1H-pyrrol-1-yl)propanamide
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
3-{2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-(2-methoxyphenoxy)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
7-(5-chloro-2-methoxyphenyl)-4-(1H-indol-2-ylmethyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-N-cyclopentyl-N-[2-(dimethylamino)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(2-hydroxy-3-{4-[(3-hydroxyazetidin-1-yl)methyl]-2-methoxyphenoxy}propyl)piperidin-4-ol
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-[(3-methyloxetan-3-yl)methyl]acetamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}dimethylamine
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(3-phenyl-1,2-oxazole-5-carbonyl)-4-propyl-1,4-diazepan-5-one
1-[2-(4-methoxyphenyl)ethyl]-5-(5-oxopyrrolidine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxylate
1-(5-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(3R,4R)-1-[2-(methylsulfanyl)benzoyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-(methoxymethyl)-5-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1,2-oxazole-3-carboxamide
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(4-methylphenoxy)piperidine-4-carboxylic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
6,7-dimethoxy-2-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(4aS,8aR)-1-(3-aminopropyl)-6-{thieno[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
(2S)-2-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}-2-phenylethan-1-ol
3-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-3-yl}benzoic acid
4-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]-1-(oxolan-2-ylmethyl)piperidine
3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
methyl 6-[(2,5-dimethylphenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine
1-(propan-2-yl)-4-(pyridin-3-ylmethyl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
3-(diethylamino)-1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-cyclooctyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-{methyl[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}propan-1-ol
1-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
4-{1-[(4-methylpiperazin-1-yl)sulfonyl]piperidin-3-yl}benzoic acid
2-[3,5-dimethyl-4-(pyrimidin-5-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)propanamide
2,6-dimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrimidine-4-carboxamide