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2-(5-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-[2-(5-chloro-6-methyl-1-benzofuran-3-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-N-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
2-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
1-(4-methoxyphenyl)-4-[(5-propylfuran-2-yl)methyl]piperazin-2-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-phenoxypropan-1-one
(2R)-2-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)formamido]propanamide
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
1-benzyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1H-pyrazole-4-carboxamide
4-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-1-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
3-{[(furan-3-ylmethyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-{5-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
2-amino-1-{6-methyl-5-[5-(1-methylpyrrolidin-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
N3-ethyl-4-oxo-1-(2-phenylethyl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}piperidin-2-one
4-methyl-9-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
6-[(diethylamino)methyl]-N-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[(3-fluorophenyl)methyl]-1-(furan-2-carbonyl)-1,4-diazepan-5-one
N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}pyridine-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(1-methoxy-2-methylpropan-2-yl)-N-methylbenzamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1H-1,3-benzodiazole-7-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][1-(3-fluorophenyl)propan-2-yl]amine
N-(2,5-dimethoxyphenyl)-4-methoxy-4-phenylpiperidine-1-carboxamide
1-(1H-indazol-6-yl)-5-methyl-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperazin-2-one
6-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(4-hydroxypiperidin-1-yl)acetamide
2-(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}azetidin-3-yl)pyridine
1-{2-[(5-methyl-2-phenyl-1H-imidazol-4-yl)formamido]ethyl}piperidine-3-carboxamide
1-{2-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
(3R,4R)-3,4-dimethyl-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-3-ol
(3aR,6aR)-2-cyclobutanecarbonyl-5-(3-methoxy-4-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-methylbut-2-en-1-yl)-1-(1,3-thiazole-4-carbonyl)piperidine-3-carboxylic acid
5-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]-4,5,6,7-tetrahydro-1H-indazole
({2-methoxy-5-[4-phenyl-1-(prop-2-yn-1-yl)-1H-imidazol-5-yl]phenyl}methyl)dimethylamine
2-[4-(6-aminopyridine-3-carbonyl)morpholin-3-yl]-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[3-(1H-pyrazol-4-yl)phenyl]methyl}amine
3-{5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
6-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazin-2-amine
7-(propan-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(4-hydroxypiperidin-1-yl)ethyl]acetamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(thiophen-3-ylmethyl)amine
N-(2,2-dimethyloxan-4-yl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(4-propanoylphenoxy)acetamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(6-methylpyridin-2-yl)methyl](oxolan-2-ylmethyl)amine
2-(4-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}piperazin-1-yl)pyrimidine
2-acetyl-8-[(2,6-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid