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1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(thian-4-yl)piperazine
(1S)-3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-phenylpropan-1-ol
1-[(2S)-2-[1-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-1-yl]propan-1-one
3-[5-(1H-imidazol-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-methyl-1,2-dihydroquinolin-2-one
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-cyclopentyl-2-phenylethyl)-1,1-dioxo-1λ6-thiane-4-carboxamide
4-[3-(dimethylamino)pyrrolidin-1-yl]-N,N,5,6-tetramethylpyrimidin-2-amine
N-(2,3-dihydro-1H-inden-1-yl)-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
2-[2-({[2-(azepan-1-yl)ethyl](propan-2-yl)amino}methyl)phenoxy]acetic acid
(3aS,6aS)-2-(ethanesulfonyl)-5-(quinoxalin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
1-(azocan-1-yl)-3-[5-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-(5-fluoro-2-methylphenyl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
ethyl 2-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)amino]acetate
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]urea
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
1-({[1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
(2S,4R)-1-(2-ethoxyacetyl)-N-ethyl-4-[2-(3-hydroxyphenyl)acetamido]pyrrolidine-2-carboxamide
1-({1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}methyl)-4-methylpiperazine
6-ethyl-N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(morpholin-4-yl)pyrimidin-4-amine
3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
7-(1-benzothiophen-3-yl)-9-methoxy-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
4-[2-(carbamoylmethoxy)-5-methylphenyl]-N,N-dimethylbenzamide
4-methyl-6-[4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperazin-1-yl]pyrimidin-2-amine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)pyrrolidine-1-carboxamide
(3S,4R)-1-[3-(1H-imidazol-2-yl)benzoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-[1-(5-chloropyridine-2-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
8-{1H-pyrrolo[2,3-b]pyridin-6-yl}-2,8-diazaspiro[4.5]decan-3-one
1-cyclopropanecarbonyl-4-{4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenoxy}piperidine
8-(3-aminobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-[3-(4-methoxyphenyl)-3-phenylpropanoyl]piperazin-2-one
1-(2-methylpropyl)-3-(4-phenylazepane-1-carbonyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
4-(1H-1,2,4-triazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)butan-1-one
5-(methoxymethyl)-N-[1-(thian-4-yl)piperidin-4-yl]thiophene-2-carboxamide
7-(cyclopropylmethyl)-2-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}morpholin-3-yl)-N-(pyridin-3-ylmethyl)acetamide
N-methyl-5-[2-(1H-pyrazol-1-yl)butanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
(3R,4R)-3-methyl-1-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-4-(oxan-4-yl)piperidin-4-ol
1-[(3-chloro-1H-indol-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
4-[3-(1H-pyrazol-1-yl)phenyl]-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(4S)-1-(4-chloro-2-hydroxybenzoyl)-3,3,4-trimethylpiperidin-4-ol
1,7-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2,4-dioxo-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-5-carboxamide
1-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-3-(5-methyl-4H-1,2,4-triazol-3-yl)urea
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
2-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)pyridine
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide