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2-amino-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(1R,5R)-N,N-dimethyl-6-[2-(pyridin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(4-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)piperidin-4-ol
3-chloro-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-fluoro-1-benzothiophene-2-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
1-(4-methylpyrimidine-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
2-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-chlorophenoxy)propanoic acid
3-[(4-{[(1-cyclopropyl-1H-imidazol-5-yl)methyl]amino}-6-methylpyrimidin-2-yl)amino]phenol
N-(1-methoxy-2-methylpropan-2-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(2-methylpropyl)-8-[6-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-butanoyl-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-4-cyclopropyl-1-[3-(2-fluorophenyl)propanoyl]pyrrolidine-3-carboxylic acid
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(oxolan-2-ylmethyl)piperidin-4-amine
1-(2-methoxyphenyl)-4-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
[(3R,4S)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-[2-(prop-2-en-1-yloxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[1-(4-methylphenyl)propyl]-1,2-oxazole-3-carboxamide
3-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
4-[1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]benzoic acid
4-{1-[4-(2-methoxyphenyl)benzoyl]azetidin-3-yl}pyridine
2-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}pyridine-3-carboxamide
3-{1-[(2,3-dimethoxyphenyl)methyl]-4-phenyl-1H-imidazol-5-yl}pyridine
2-(dimethylamino)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-2-(2-methylphenyl)acetamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-ylmethyl}-1,2,4-oxadiazole-5-carboxamide
1-(2-fluorophenyl)-N-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)piperidin-4-amine
3,5-dimethoxy-N-({1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methyl)benzamide
2-(2-methyl-1-benzofuran-5-carbonyl)-2,3-dihydro-1H-isoindole
2-(2-butoxy-5-methylphenyl)-2-(4-hydroxypiperidin-1-yl)acetic acid
1-(3-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
(5S,9aS,9bS)-5-[5-(hydroxymethyl)furan-2-yl]-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3,4,7-trimethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
1-(2-aminoethyl)-N-[(4-phenylmorpholin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-1,2,3-triazol-4-yl)piperidine
4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]pyrimidine
1-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethyl-N-(2-phenylethyl)pyrrolidine-3-carboxamide
3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-(thiophen-3-ylmethyl)piperidine
[4-benzyl-1-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-yl]methanol
1-ethyl-8-{[2-(furan-2-yl)phenyl]methyl}-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
dimethyl(2-{[(2-methylphenyl)methyl](oxolan-3-ylmethyl)amino}ethyl)amine
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
(1R,2S,6R,7S)-4-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-azatricyclo[5.2.2.02,6]undecane
2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
methyl 3-({[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate