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4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(pyridin-3-yloxy)propyl]benzamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
[1-(4-aminopyrimidin-2-yl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4,6-dimethyl-2-oxo-2H-pyran-5-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3-fluoropyridine-4-carboxamide
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}isoquinoline
2-(2-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
ethyl 3-[(1,3-benzothiazol-2-yl)amino]azepane-1-carboxylate
2-[methyl(2-phenylethyl)amino]-N-[(1s,4s)-4-aminocyclohexyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 5-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-2,4-dimethyl-1H-pyrrole-3-carboxylate
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-3-carbonitrile
2-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyrimidine
8-(1H-indole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-ethyl-8-[(1-methyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
dimethyl(2-{[(2-methylphenyl)methyl]({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})amino}ethyl)amine
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]quinoline-8-sulfonamide
{[1-({1-[(1-methyl-1H-pyrrol-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl}urea
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]propanamide
1-(carbamoylmethyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
methyl 3-({[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)propanoate
2-(4-fluorophenyl)-4-[5-(methanesulfonylmethyl)pyridin-2-yl]morpholine
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(ethylamino)pyrimidine-5-carboxamide
1-(3-{[3-(4H-1,2,4-triazol-4-yl)phenyl]formamido}propyl)piperidine-3-carboxamide
N-(2-{4-phenyl-5-[6-(trifluoromethyl)pyridin-3-yl]-1H-imidazol-1-yl}ethyl)acetamide
4-[2-(pyridin-4-yl)quinoline-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
3-(4-chloro-2-methylbenzoyl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine
5-(oxolan-2-yl)-N-[2-(pyridin-2-yl)ethyl]thiophene-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}propanamide
N-[2-(1H-indol-1-yl)ethyl]-N,2-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-(1,4-dioxan-2-ylmethyl)-2-(propan-2-yl)-1H-imidazole
6-{1,4-dioxa-8-azaspiro[4.5]decan-8-yl}-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-phenylbutanamide
4-(1-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidin-3-yl)morpholine
1-{2-methoxy-5-[(4-propylpiperazin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
4-(5-methylfuran-2-yl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
(1S,6R)-3-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
3-cyclopropyl-1-(2,3-dihydro-1H-inden-5-yl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
1-methyl-3-(4-phenoxyphenyl)-4-[(2-phenylazetidin-1-yl)methyl]-1H-pyrazole
(3R)-3,4,4-trimethyl-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-propylcyclopropyl)-1,3-oxazole-4-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
5-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
dimethyl(2-{4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]morpholin-2-yl}ethyl)amine
4-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-4H-1,2,4-triazole
3-[1-(cyclohexylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]propanoic acid
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide