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3-[(3R,4S)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
5-[3-chloro-4-(pyrrolidin-1-yl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(1S,5R)-6-(5-cyclopropyl-1H-pyrazole-3-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}pyridin-3-ol
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-2-ylmethyl)piperazine
N5-methyl-N5-(oxolan-3-yl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(4-methyl-1H-imidazole-2-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(morpholin-4-yl)-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
N-(2-methoxyethyl)-1-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-4-yl}piperidine-3-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-[(2R)-pyrrolidine-2-carbonyl]piperidine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenylprop-2-ynamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyridin-2-amine
(4aS,8aR)-6-(3-hydroxypropanoyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-(2-methoxybenzoyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
4-(2-methoxyphenoxy)-1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidine
3-(2,5-difluorobenzoyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-methyl-N-[2-(2-methylphenyl)-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}ethyl]cyclobutanecarboxamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
[1-(1H-1,3-benzodiazol-2-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
4-[1-(2-ethylbenzoyl)piperazine-2-carbonyl]morpholine
6,8-dimethyl-2-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
1-cyclopentyl-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[methyl(phenyl)amino]ethan-1-one
3-{3-cyclopropyl-5-[2-(1H-imidazol-2-yl)phenyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
4-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}benzoic acid
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidin-2-amine
3-({2-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(4-tert-butylphenyl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
3-phenyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
1-(4-chlorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
N-[2-(dimethylamino)ethyl]-3,4-difluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
N-butyl-N-(furan-2-ylmethyl)-2-(phenylformamido)acetamide
1-[1-(2-methylpropanoyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-phenoxy-5-[2-(propan-2-yl)-1H-imidazol-1-yl]pyridine
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
1-[1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-1H-imidazole-5-carboxamide
3-{[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]methyl}benzoic acid
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
methyl 6-[(4-fluoro-3-methoxyphenyl)methyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(3-fluoropyridin-2-yl)-1H-pyrazol-1-yl]acetamide
(1S,5R)-3-(pyridin-4-ylmethyl)-6-{[4-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2,5-dimethyl-3-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]pyrazine
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2-(pyridin-3-yl)pyrimidine