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N-[1-(cyclohex-1-en-1-yl)ethyl]-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
(3S)-1,3-dimethyl-4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
1-(2-methoxyethyl)-5-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
6-ethyl-4-{[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2H-chromen-2-one
[(5-ethylpyridin-2-yl)methyl]({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)methylamine
2-{4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
3-[(2R,3R,6R)-5-(1H-1,3-benzodiazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-(diphenylmethyl)-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
methyl 4-{[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-{[2-ethyl-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
1-methyl-4-{thieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
[5-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)furan-2-yl]methanol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}(naphthalen-2-ylmethyl)amine
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(2-phenoxyethyl)piperazine
N-(1-benzothiophen-2-ylmethyl)-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,2,6-trimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-methyl-3-[({[4-(methylsulfanyl)phenyl]methyl}(propyl)amino)methyl]pyridin-2-amine
2-(2-hydroxyethyl)-9-[2-(methylsulfanyl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-(adamantan-1-yl)-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[2-(benzyloxy)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
2,6-dimethyl-5-(2-oxo-2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
4-chloro-N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
3-[2-(2,2-dimethyl-3-oxopiperazin-1-yl)-2-oxoethyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(3S,4R)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-[methyl(phenyl)amino]-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2-hydroxybenzoate
3-benzyl-1-methyl-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{5-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]thiophen-2-yl}ethan-1-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethylthiophene-3-carboxamide
3-({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
(4aS,8aR)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N,N-dimethyl-1-{[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-3-amine
2-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
8-[3-(1H-imidazol-1-yl)propyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-[(2R,3R,6R)-5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]phenoxy}acetic acid
4-(1H-pyrazol-3-yl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-({[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]carbamoyl}amino)ethyl]acetamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[2-(1,4-diazepan-1-ylmethyl)phenyl]-6-(phenoxymethyl)-3,4-dihydropyrimidin-4-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)azepane-4-carboxamide
2-({2-oxo-1,3-dioxa-8-azaspiro[4.5]decan-8-yl}methyl)benzonitrile
1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}-2-phenylethan-1-one
3-[3-cyclopentyl-5-(2-methoxy-4-methylphenyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
2-(cyclobutylmethyl)-6,7-dimethoxyquinazolin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}pent-4-enamide