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3-{[(2,6-dimethylphenyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
4-cyano-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
2-(2,5-dimethylphenoxy)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)propanamide
5-(1-{[4-(1,2,3-thiadiazol-4-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
1-amino-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]cyclopropane-1-carboxamide
4-({1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}amino)pyrimidine-5-carboxylic acid
ethyl 1-{[7-fluoro-2-oxo-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperidine-3-carboxylate
3-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)benzoic acid
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
6-(4-fluorophenyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-methanesulfonyl-1'-{spiro[2.3]hexane-1-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-hydroxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
2-[2-(2-methylbutyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
2-{1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-5-methyl-1H-1,3-benzodiazole
6-methyl-5-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
dimethyl[3-(2-{1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
2-[4-(ethylsulfanyl)phenyl]-2-{methyl[(3-methylpyridin-4-yl)methyl]amino}acetic acid
N-methyl-N-[4-(morpholin-4-yl)butyl]-1H-pyrazole-4-carboxamide
2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-5-methoxyphenol
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(2-ethylphenoxy)azetidine
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
[9-(4-aminopyrimidin-2-yl)-3-(2-ethoxyethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-(3-chlorophenyl)-4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-5-methylpiperazin-2-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[4-(2-methylphenyl)phenyl]methyl}piperidine
1-cyclohexyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}piperidine-4-carboxamide
2-methyl-4-(piperidin-4-yl)-6-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrimidine
4-(2-chloro-4-fluorophenyl)-3-ethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-N-[(3-chlorophenyl)methyl]propanamide
6-[4-(1-methylazepane-2-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
(2S,4R)-N-(2-methoxyethyl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-{4-[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)propan-1-ol
3-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-imidazol-2-yl}phenol
4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)-N-[4-(propan-2-yl)phenyl]piperazine-1-carboxamide
4-benzyl-3-{1-[2-(pyridin-3-yloxy)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
4-ethyl-3-{1-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]propanamide
methyl 4-{[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]methyl}benzoate
2-(benzylsulfanyl)-N4-[2-(1H-pyrazol-4-yl)ethyl]pyrimidine-4,6-diamine
N-[(5-methylpyrazin-2-yl)methyl]-1,3-diphenyl-1H-pyrazole-5-carboxamide
2-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
6-[1-(thiophen-2-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1S,5R)-3-[2-(4-acetylphenoxy)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one