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(4aS,7aR)-1-[4-(1H-imidazol-1-yl)butanoyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-methylbutyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-benzyl-4-(3-fluoropyridin-2-yl)-1,4-diazepan-6-ol
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,4-dimethyl-1,3-oxazole-5-carboxamide
3-{4-phenyl-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}propan-1-ol
2-(5-methyl-1,2-oxazol-3-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
2,3-dimethoxy-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N,N-dimethyl-2-({[methyl(propan-2-yl)sulfamoyl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-{[cyclopropyl(thiophen-3-ylmethyl)amino]methyl}-6-methyl-1,2-dihydroquinolin-2-one
2-{8-[(2,3-difluorophenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
(1S,4S)-2-(2-methoxy-5-methylphenyl)-5-[(2E)-2-methylbut-2-en-1-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-{[methyl({[1-(propan-2-yl)piperidin-3-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-[1-({1-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]pyridine
8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-ethyl-2-methyl-4-[4-(oxan-4-yl)piperazin-1-yl]pyrimidine
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-[2-(propan-2-yl)phenyl]piperidine-1-carboxamide
4-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridin-2-amine
N-[3-(cyclopentyloxy)propyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepan-6-ol
3-ethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-indole-2-carboxamide
3-{[2-(dimethylamino)-2-(2-methylphenyl)acetamido]methyl}-N,N-dimethylbenzamide
[1-(azepane-1-sulfonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
(1R,5R)-6-[(6-methylpyridin-2-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-acetamidopropanamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(4-hydroxypiperidin-1-yl)acetamide
(1s,4s)-4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
(2S)-2-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]-2-phenylacetamide
2-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(thiophen-2-ylmethyl)amino]ethan-1-ol
9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
5-cyclopropanecarbonyl-1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(morpholin-4-yl)acetamide
2-{4-[(6-chloroquinolin-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-(2-fluoroethyl)-9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-[5-(2,3-dihydro-1H-inden-2-yl)-1,2,4-oxadiazol-3-yl]pyrazine
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
4-(2,5-dimethylthiophen-3-yl)-2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-(methoxymethyl)-1H-pyrazol-1-yl}pyrimidine
N-cyclopropyl-3-(ethanesulfinyl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
2-ethyl-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
3-cyclopropyl-1-(3,4-dimethylphenyl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
2-phenyl-1-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}ethan-1-ol