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2-[2-(dimethylamino)ethyl]-9-(5,6-dimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[2-(furan-2-yl)azepan-1-yl]methyl}pyridin-2-amine
6-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-2-carbonitrile
methyl 1-methoxy-2-oxo-8-(5-phenyl-1,2-oxazole-3-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
2-{5-[1-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
1-{1-[4-(2-methoxyethyl)piperidin-1-yl]propan-2-yl}-1H-1,3-benzodiazole
(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-5-[2-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(pyrazin-2-yl)-2-{[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amino}acetamide
N-[3-(1H-imidazol-1-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(2,3-dihydro-1H-inden-4-yl)-3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)urea
2-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,2,3-trimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-({5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
5-ethyl-2-methyl-4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidine
(4aS,7aR)-1-[2-(2-methoxyphenoxy)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5,8-dimethyl-2-({[3-(4H-1,2,4-triazol-4-yl)propyl]amino}methyl)quinolin-4-ol
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-3-(quinoxalin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(3S,4S)-3-hydroxy-4-[methyl(propyl)amino]pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carbonyl]azepane
4-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
{3-[2-(2,6-difluorophenyl)-1H-imidazol-1-yl]propyl}dimethylamine
1-(2-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(1-{1-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]propan-2-yl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-[2-(2-methoxyphenyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[1-(thiophen-3-yl)propan-2-yl]-3,4-dihydropteridin-4-one
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
3-{[1-(1H-indol-2-yl)ethyl](methyl)amino}-N-(1,3-thiazol-2-yl)propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(1R,5R)-6-methyl-3-(3-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-1-yl}pyrimidine
9-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-(hydroxymethyl)-1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
2-(dimethyl-1,3-thiazol-4-yl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}acetamide
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(3,5-difluoro-2-methoxyphenyl)-2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}acetic acid
1-[(3,4-difluorophenyl)methyl]-3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
3-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidin-2-one
N-[2-(dimethylamino)ethyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
6-ethyl-2-oxo-N-(piperidin-3-ylmethyl)-1,2-dihydropyridine-4-carboxamide
8-(2-propyl-1,3-thiazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,3-thiazole-5-carboxamide
N-[2-(2-fluorophenyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
N-(1,3-dihydro-2-benzofuran-5-yl)-4-(2-methoxyphenyl)piperidine-1-carboxamide
N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
(3R,4S)-4-cyclopropyl-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-3-amine