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N-(4-fluorophenyl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
1-(4-{[(5-methylpyrazin-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[3-(4-ethyl-2-methyl-3-oxopiperazin-1-yl)-3-oxopropyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-cyclobutyl-5-fluoro-1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
methyl 3-{[(2-fluorophenyl)formamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
4-[(2-ethoxyphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
N-(2,4-dimethylphenyl)-3-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]propanamide
1-(6-methylpyridin-2-yl)-4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazine
N-cyclopentyl-1-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(furan-2-ylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(4aS,8aS)-2-{[2-(2-hydroxyethoxy)phenyl]methyl}-decahydroisoquinolin-4a-ol
N-butyl-3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propanamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
1-(methoxymethyl)-N-[2-(4-sulfamoylphenyl)ethyl]cyclobutane-1-carboxamide
5-(2-chlorophenyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}furan-2-carboxamide
2-ethyl-N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-5-carboxamide
4-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-(3-fluorophenyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzoxazole-5-carboxamide
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2,6-trimethylquinoline-4-carboxamide
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(furan-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(1-ethylpiperidin-4-yl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methyl-5-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1,7-dimethyl-2-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1H-indole
4-[(4-hydroxypiperidin-1-yl)methyl]-N-(4-methoxy-3,5-dimethylphenyl)benzamide
N-[(2S,4R,6R)-2-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-6-cyclohexyloxan-4-yl]acetamide
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-(cyclopropylmethyl)-N-methyl-5-(3-phenylprop-2-ynoyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(3-chlorophenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}-2-(3-propoxyphenyl)acetic acid
9-(2-hydroxyethyl)-1-methyl-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-(3,4-dimethoxyphenyl)piperidin-3-amine
(2S,4R)-4-amino-N,N-diethyl-1-(morpholine-4-sulfonyl)pyrrolidine-2-carboxamide
2-(2-hydroxypropyl)-9-(2-methylfuran-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(3-methoxyphenyl)piperidine-1-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-chloro-4-fluorophenoxymethyl)-4-(pyrrolidine-1-carbonyl)-1,3-oxazole
3-(3-fluoropyridin-4-yl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
(3aR,6aS)-5-(1-benzofuran-2-ylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-2-(2-{[2-(6-methylpyridin-2-yl)ethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
4-(4-chloro-2-hydroxybenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-4-(4-methylpiperazin-1-yl)pentanamide
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)cyclopropanesulfonamide
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine