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1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3-(hydroxymethyl)piperidin-3-ol
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidine-3-carboxamide
1-(3,4-difluorophenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
(3R)-1-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-ol
ethyl 5-{[(5-methylpyrazin-2-yl)methyl]carbamoyl}-1H-imidazole-4-carboxylate
3-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-1-[3-(4-methylpiperazin-1-yl)propyl]urea
3-(propan-2-yl)-1-{2-[1-(3,3,3-trifluoropropyl)piperidin-3-yl]ethyl}urea
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-1,3-thiazole-5-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
{2-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}urea
5-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-methyl-1,2,4-oxadiazole
1-methyl-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-1,4-dihydroquinolin-4-one
1-[(2,4-difluorophenyl)methyl]-4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}piperidin-4-ol
2-methoxy-1-[1'-(3-methylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
2-(3-acetylphenyl)-N-propylbenzamide
(1R,5R)-6-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3S,4R)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-(3,3-diphenylpiperidin-1-yl)-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-methyl-6-oxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
1,3,6-trimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(3-methyl-1H-pyrazol-1-yl)-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}propanamide
[5-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
N-methyl-3-[(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)sulfamoyl]benzamide
(2S)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-3-phenylpropan-1-one
4-[7-(3-cyanopyridin-2-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
7-methyl-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4H-chromen-4-one
methyl({[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl})[1-(thiophen-2-yl)ethyl]amine
1-(2-methoxyethyl)-N-[2-(naphthalen-1-yl)propan-2-yl]-6-oxopiperidine-3-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-(3-phenylbenzoyl)-7-azaspiro[3.5]nonan-1-ol
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-4-(piperidin-1-yl)butan-1-one
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
1-[2-({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
2-butyl-8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-phenylmethanesulfonyl-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2,3-dimethoxy-N-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)benzamide
(3R,4R)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-cyclohexyl-5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}pyrimidine
(2S,4R)-4-amino-N,N-diethyl-1-(quinoxalin-2-yl)pyrrolidine-2-carboxamide
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-(trifluoromethyl)piperidine
(2S,4S)-4-(4-chlorobenzamido)-N,1-dimethyl-N-(1,2-oxazol-3-ylmethyl)pyrrolidine-2-carboxamide
3-hydroxy-3-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-1-(3-phenylpropyl)piperidin-2-one
3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-[3-(pyridin-2-yl)propyl]urea
[(3R,4R)-1-(3-chloro-4-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol