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(3R,4R)-1-(2-chlorobenzoyl)-3,4-dimethylpyrrolidin-3-ol
2-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-methyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-[1,2,4]triazolo[1,5-a]pyridine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-1,3-thiazole-5-carboxamide
1-{1-[3-(difluoromethoxy)benzoyl]piperidin-4-yl}-3-methylbutan-1-ol
2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N-(propan-2-yl)acetamide
methyl 6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-ethynyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzamide
N-[(3,4-difluorophenyl)methyl]-1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(azocan-1-yl)-3-[2-methoxy-4-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(3-methoxypropyl)-9-(1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(1H-pyrazol-1-yl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 1-(1H-indol-3-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-(2-ethoxyphenyl)-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
1-[4-(furan-2-yl)butan-2-yl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
2-(dimethyl-1,2-oxazol-4-yl)-2-(thiomorpholin-4-yl)acetic acid
1-(3-chlorophenyl)-4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-5-methylpiperazin-2-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxamide
N-(4-{[(1-fluoro-3-phenylpropan-2-yl)carbamoyl]methoxy}phenyl)propanamide
2-(1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
3-(5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}furan-2-yl)-1H-pyrazole
3,5-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1-benzofuran-2-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-6-(2-aminoethyl)-2-methylpyrimidin-4-amine
2-({1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
N-[(2,5-difluorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(3-{[1-(2,3,6-trimethylquinoline-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-[(1-methyl-1H-indol-2-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-cyclobutanecarbonyl-6-methyl-5-[5-(1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
methyl[(4-methylphenyl)methyl][(2,3,4-trimethoxyphenyl)methyl]amine
N-[1-(2,5-difluorophenyl)cyclopropyl]-4-(1H-pyrazol-3-yl)benzamide
1-(2-methoxyacetyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
N'-(2,3-dimethylphenyl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)propanediamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(3E)-hex-3-enoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanoic acid
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
4-ethyl-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2S)-1-oxo-1-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]propan-2-yl]acetamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
2-(4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)acetamide
5-methyl-3-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole-2-carboxylic acid
5-{2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
N-methyl-5-{[2-(2-phenylethyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
2,6-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
N-ethyl-2-(1-methyl-1H-pyrrol-2-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxoacetamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(2,5-dimethoxyphenyl)pyridine-3-carbonitrile
4-(5-amino-1H-pyrazole-3-carbonyl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one