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butyl 9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxylate
ethyl 3-[(3-chlorophenyl)methyl]-1-(2-methylfuran-3-carbonyl)piperidine-3-carboxylate
9-(2-hydroxyacetyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[3-(2-hydroxyethyl)-4-methylpiperazine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
2-[5-(2-phenoxyethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
(1S,6R)-9-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(3aR,6aS)-2-(2,3-dihydro-1H-indene-1-carbonyl)-octahydropyrrolo[3,4-c]pyrrole
(3S,9aR)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-2-ylsulfanyl)acetamide
4-({4-methyl-5-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyridine
6-fluoro-2-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-ylmethyl)quinolin-4-ol
5-acetyl-2,4-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrrole-3-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyrrolidin-1-yl)butan-1-one
N-(2H-1,3-benzodioxol-5-yl)-5-(1-benzyl-4-hydroxypiperidin-4-yl)-1-benzofuran-2-carboxamide
2-[5-(methylcarbamoyl)thiophen-2-yl]-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)pyrrolidine-1-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
1-(2-chlorobenzoyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-benzotriazole
3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(1S,4S)-2-(2-fluorophenyl)-5-[4-(trifluoromethyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-7-methoxy-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
N-cyclopropyl-1-[2-(methylamino)pyridine-3-carbonyl]piperazine-2-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[4-(dimethylamino)phenyl]acetamide
[(2,3-difluorophenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-(4-{1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}piperidin-1-yl)ethan-1-one
1-[(4,5-dimethylfuran-2-yl)methyl]-4-[(4-fluorophenyl)methyl]-1,4-diazepane
1-({6-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridin-3-yl}methyl)-4-methylpiperazine
1-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
(4aR,7aS)-1-(2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxy-4-(prop-2-en-1-yl)piperidine
N'-(4-methylphenyl)-N-[(1-propylcyclobutyl)methyl]propanediamide
ethyl 4-{[4-(propylsulfanyl)phenyl]carbamoyl}piperazine-1-carboxylate
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-methyl-5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenol
6-(5-fluoro-2-methoxyphenyl)pyrazine-2-carboxamide
1-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-4-(benzyloxy)butan-1-one
3-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-[4-(4-methylphenyl)phenyl]-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
2-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
3-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}quinoline
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(2,2,2-trifluoroethyl)propanamide
5-(4-tert-butylcyclohexyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]piperidine-4-carboxamide
4-chloro-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]aniline
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(methylamino)-1,3-thiazole-4-carboxamide